C-attached aminoalkylindoles: Potent cannabinoid mimetics

被引：20

作者：

DAmbra, TE

Eissenstat, MA

Abt, J

Ackerman, JH

Bacon, ER

Bell, MR

Carabateas, PM

Josef, KA

Kumar, V

Weaver, JD

Arnold, R

Casiano, FM

Chippari, SM

Haycock, DA

Kuster, JE

Luttinger, DA

Stevenson, JI

Ward, SJ

Hill, WA

Khanolkar, A

Makriyannis, A

机构：

[1] SANOFI WINTHROP INC,DEPT MED CHEM,COLLEGEVILLE,PA 19426

[2] SANOFI WINTHROP INC,DEPT NEUROSCI,COLLEGEVILLE,PA 19426

[3] SANOFI WINTHROP INC,SANOFI RES DIV,COLLEGEVILLE,PA 19426

[4] UNIV CONNECTICUT,SCH PHARM,STORRS,CT 06269

来源：

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 1996年 / 6卷 / 01期

关键词：

D O I：

10.1016/0960-894X(95)00560-G

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

Aminoalkylindoles (AAIs) with potent cannabinoid agonist activity have been synthesized where the aminoalkyl chain is attached to the indole ring via a carbon atom of the cyclic amine.

引用

页码：17 / 22

页数：6

共 21 条

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