Soluble polymer-supported convergent parallel library synthesis

被引:29
作者
Ahn, JM
Wentworth, P
Janda, KD
机构
[1] Scripps Res Inst, Dept Chem, La Jolla, CA 92037 USA
[2] Skaggs Inst Chem Biol, La Jolla, CA 92037 USA
关键词
D O I
10.1039/b210696e
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
Soluble polymer-supported convergent synthesis has for the first time been successfully exploited for parallel library synthesis; sub-libraries of tripeptide iodoarenes and arylboronic acids reacted smoothly in a multipolymer Pd-II-catalyzed Suzuki coupling reaction to generate a library of bisaryl-linked hexapeptides.
引用
收藏
页码:480 / 481
页数:2
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