Syntheses of new pyridonecarboxylic acid derivatives containing 1- or 2-naphthyl substituents at N-1 and their anti-HIV-RT activities

被引：11

作者：

Oh, YS

Cho, SH

机构：

[1] Dong Wha Pharmaceut Ind Co Ltd, Res Labs, Anyang 430010, Kyung Ki Do, South Korea

[2] Chung Ang Univ, Dept Chem, Seoul 156756, South Korea

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 1998年 / 35卷 / 01期

关键词：

D O I：

10.1002/jhet.5570350104

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A series of new pyridonecarboxylic acid derivatives containing 1- or 2-naphthyl substituents at N-1 were synthesized and their in vitro anti-HIV-RT activities were evaluated. Several compounds in this series showed better activity than Atevirdine.

引用

页码：17 / 23

页数：7

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