Three component condensations catalyzed by iodine-alumina for the synthesis of substituted 3,4-dihydropyrimidin-2(1H)-ones under microwave irradiation and solvent-free conditions

被引：67

作者：

Saxena, I ^{[1
]}

Borah, DC ^{[1
]}

Sarma, JC ^{[1
]}

机构：

[1] Reg Res Lab, Natl Prod Chem Div, Jorhat 785006, Assam, India

来源：

TETRAHEDRON LETTERS | 2005年 / 46卷 / 07期

关键词：

D O I：

10.1016/j.tetlet.2004.12.081

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Condensation of an aldehyde, ethyl acetoacetate and urea or thiourea under microwave irradiation in the presence of 10% iodine adsorbed on neutral alumina gives substituted 3,4-dihydropyrimidin-2(1H)-ones in excellent yields. (C) 2004 Elsevier Ltd. All rights reserved.

引用

页码：1159 / 1160

页数：2

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