Solid-phase synthesis of 2-aminothiazoles

被引：156

作者：

Kearney, PC ^{[1
]}

Fernandez, M ^{[1
]}

Flygare, JA ^{[1
]}

机构：

[1] Tularik Inc, S San Francisco, CA 94080 USA

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1998年 / 63卷 / 01期

关键词：

D O I：

10.1021/jo971542a

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

[No abstract available]

引用

页码：196 / 200

页数：5

共 24 条

[1]

[Anonymous], ANGEW CHEM INT EDIT, DOI DOI 10.1002/ANIE.199622881

[2] A convenient procedure for the solution phase preparation of 2-aminothiazole combinatorial libraries [J].

Bailey, N ;

Dean, AW ;

Judd, DB ;

Middlemiss, D ;

Storer, R ;

Watson, SP .

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1996, 6 (12) :1409-1414

[3] PHENETHYLTHIAZOLETHIOUREA (PETT) COMPOUNDS, A NEW CLASS OF HIV-1 REVERSE-TRANSCRIPTASE INHIBITORS .1. SYNTHESIS AND BASIC STRUCTURE-ACTIVITY RELATIONSHIP STUDIES OF PETT ANALOGS [J].

BELL, FW ;

CANTRELL, AS ;

HOGBERG, M ;

JASKUNAS, SR ;

JOHANSSON, NG ;

JORDAN, CL ;

KINNICK, MD ;

LIND, P ;

MORIN, JM ;

NOREEN, R ;

OBERG, B ;

PALKOWITZ, JA ;

PARRISH, CA ;

PRANC, P ;

SAHLBERG, C ;

TERNANSKY, RJ ;

VASILEFF, RT ;

VRANG, L ;

WEST, SJ ;

ZHANG, H ;

ZHOU, XX .

JOURNAL OF MEDICINAL CHEMISTRY, 1995, 38 (25) :4929-4936

[4] Solid-phase synthesis of 1,4-benzodiazepine-2,5-diones. Library preparation and demonstration of synthesis generality [J].

Boojamra, CG ;

Burow, KM ;

Thompson, LA ;

Ellman, JA .

JOURNAL OF ORGANIC CHEMISTRY, 1997, 62 (05) :1240-1256

[5] 4-HYDROXY-3-QUINOLINECARBOXAMIDES WITH ANTIARTHRITIC AND ANALGESIC ACTIVITIES [J].

CLEMENCE, F ;

LEMARTRET, O ;

DELEVALLEE, F ;

BENZONI, J ;

JOUANEN, A ;

JOUQUEY, S ;

MOUREN, M ;

DERAEDT, R .

JOURNAL OF MEDICINAL CHEMISTRY, 1988, 31 (07) :1453-1462

[6]

DROBNICA L, 1977, CHEM CYANATES THEI 2, P1109

[7] Design, synthesis, and evaluation of small-molecule libraries [J].

Ellman, JA .

ACCOUNTS OF CHEMICAL RESEARCH, 1996, 29 (03) :132-143

[8] REDUCTIVE ALKYLATION ON A SOLID-PHASE - SYNTHESIS OF A PIPERAZINEDIONE COMBINATORIAL LIBRARY [J].

GORDON, DW ;

STEELE, J .

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1995, 5 (01) :47-50

[9]

GREENE TW, 1991, PROTECTIVE GROUPS OR

[10]

Hantzsch A, 1887, CHEM BER, V20, P3118, DOI [10.1002/cber.188702002200, DOI 10.1002/CBER.188702002200]

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