An improved synthesis of substituted benzolblthiophenes using microwave irradiation

被引:22
作者
Allen, D [1 ]
Callaghan, O [1 ]
Cordier, FL [1 ]
Dobson, DR [1 ]
Harris, JR [1 ]
Hotten, TM [1 ]
Owton, WM [1 ]
Rathmell, RE [1 ]
Wood, VA [1 ]
机构
[1] Eli Lilly & Co, Lilly Res Ctr, Windlesham GU20 6PH, Surrey, England
关键词
benzothiophenes; cyclisation; decarboxylation; microwave irradiation;
D O I
10.1016/j.tetlet.2004.11.005
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
An easy and high-yielding method for the synthesis of substituted benzo[b]thiophenes using microwave irradiation is described. (C) 2004 Elsevier Ltd. All rights reserved.
引用
收藏
页码:9645 / 9647
页数:3
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