BIOCHEMICAL AND PHARMACOLOGICAL CHARACTERIZATION OF AN EXTREMELY POTENT AND SELECTIVE NONPEPTIDE CHOLECYSTOKININ ANTAGONIST

被引：697

作者：

CHANG, RSL

LOTTI, VJ

机构：

来源：

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA | 1986年 / 83卷 / 13期

关键词：

D O I：

10.1073/pnas.83.13.4923

中图分类号：

O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];

学科分类号：

07 ; 0710 ; 09 ;

摘要：

引用

页码：4923 / 4926

页数：4

共 34 条

[1] SOME QUANTITATIVE USES OF DRUG ANTAGONISTS [J].

ARUNLAKSHANA, O ;

SCHILD, HO .

BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1959, 14 (01) :48-58

[2]

BENNETT JP, 1976, MOL PHARMACOL, V12, P373

[3] SPECIFIC BENZODIAZEPINE RECEPTORS IN RAT-BRAIN CHARACTERIZED BY HIGH-AFFINITY [DIAZEPAM-H-3] BINDING - (AFFINITY BINDING DIAZEPAM ANXIOLYTIC ACTIVITY BRAIN MEMBRANES REGIONAL DISTRIBUTION) [J].

BRAESTRUP, C ;

SQUIRES, RF .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1977, 74 (09) :3805-3809

[4]

BURT DR, 1976, MOL PHARMACOL, V12, P800

[5]

BYLUND DB, 1976, MOL PHARMACOL, V12, P568

[6] INCREASE IN BRAIN I-125-LABELED CHOLECYSTOKININ (CCK) RECEPTOR-BINDING FOLLOWING CHRONIC HALOPERIDOL TREATMENT, INTRACISTERNAL 6-HYDROXYDOPAMINE OR VENTRAL TEGMENTAL LESIONS [J].

CHANG, RSL ;

LOTTI, VJ ;

MARTIN, GE ;

CHEN, TB .

LIFE SCIENCES, 1983, 32 (08) :871-878

[7] NEUROPEPTIDE-Y (NPY) BINDING-SITES IN RAT-BRAIN LABELED WITH I-125 BOLTON-HUNTER NPY - COMPARATIVE POTENCIES OF VARIOUS POLYPEPTIDES ON BRAIN NPY BINDING AND BIOLOGICAL RESPONSES IN THE RAT VASDEFERENS [J].

CHANG, RSL ;

LOTTI, VJ ;

CHEN, TB ;

CERINO, DJ ;

KLING, PJ .

LIFE SCIENCES, 1985, 37 (22) :2111-2122

[8] HETEROGENEITY OF HISTAMINE H1-RECEPTORS - SPECIES VARIATIONS IN [MEPYRAMINE-H-3 BINDING OF BRAIN MEMBRANES [J].

CHANG, RSL ;

TRAN, VT ;

SNYDER, SH .

JOURNAL OF NEUROCHEMISTRY, 1979, 32 (06) :1653-1663

[9] A POTENT NONPEPTIDE CHOLECYSTOKININ ANTAGONIST SELECTIVE FOR PERIPHERAL-TISSUES ISOLATED FROM ASPERGILLUS-ALLIACEUS [J].

CHANG, RSL ;

LOTTI, VJ ;

MONAGHAN, RL ;

BIRNBAUM, J ;

STAPLEY, EO ;

GOETZ, MA ;

ALBERSSCHONBERG, G ;

PATCHETT, AA ;

LIESCH, JM ;

HENSENS, OD ;

SPRINGER, JP .

SCIENCE, 1985, 230 (4722) :177-179

[10] INACTIVATION OF ANGIOTENSIN-II RECEPTORS IN BOVINE ADRENAL-CORTEX BY DITHIOTHREITOL - FURTHER EVIDENCE FOR THE ESSENTIAL NATURE OF DISULFIDE BONDS [J].

CHANG, RSL ;

LOTTI, VJ ;

KEEGAN, ME .

BIOCHEMICAL PHARMACOLOGY, 1982, 31 (10) :1903-1906

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