AFFINITY OF MUSCARINIC RECEPTOR ANTAGONISTS FOR 3 PUTATIVE MUSCARINIC RECEPTOR-BINDING SITES

被引:82
作者
DELMENDO, RE [1 ]
MICHEL, AD [1 ]
WHITING, RL [1 ]
机构
[1] SYNTEX RES CORP,INST PHARMACOL,3401 HILLVIEW AVE,PALO ALTO,CA 94303
关键词
D O I
10.1111/j.1476-5381.1989.tb11838.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:457 / 464
页数:8
相关论文
共 28 条
[1]   COMPARISON OF AFFINITY CONSTANTS FOR MUSCARINE-SENSITIVE ACETYLCHOLINE RECEPTORS IN GUINEA-PIG ATRIAL PACEMAKER CELLS AT 29 DEGREESC AND IN ILEUM AT 29 DEGREESC AND 37 DEGREESC [J].
BARLOW, RB ;
BERRY, KJ ;
GLENTON, PAM ;
NIKOLAOU, NM ;
SOH, KS .
BRITISH JOURNAL OF PHARMACOLOGY, 1976, 58 (04) :613-620
[2]   EFFECTS OF IONS ON THE BINDING OF AGONISTS AND ANTAGONISTS TO MUSCARINIC RECEPTORS [J].
BIRDSALL, NJM ;
BURGEN, ASV ;
HULME, EC ;
WELLS, JW .
BRITISH JOURNAL OF PHARMACOLOGY, 1979, 67 (03) :371-377
[3]   ANTAGONIST DISCRIMINATION BETWEEN GANGLIONIC AND ILEAL MUSCARINIC RECEPTORS [J].
BROWN, DA ;
FORWARD, A ;
MARSH, S .
BRITISH JOURNAL OF PHARMACOLOGY, 1980, 71 (02) :362-364
[4]   THE EFFECT OF IONIC-STRENGTH ON CARDIAC MUSCARINIC RECEPTORS [J].
BURGEN, ASV .
BRITISH JOURNAL OF PHARMACOLOGY, 1986, 88 (02) :451-455
[5]  
BURGEN ASV, 1984, TIPS S, V5, P1
[6]  
CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099
[7]   [H-3]-LABELED RAUWOLSCINE AND [H-3]-LABELED YOHIMBINE BINDING TO RAT CEREBRAL AND HUMAN-PLATELET MEMBRANES - POSSIBLE HETEROGENEITY OF ALPHA-2-ADRENOCEPTORS [J].
CHEUNG, YD ;
BARNETT, DB ;
NAHORSKI, SR .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1982, 84 (1-2) :79-85
[8]   ACTION OF AGONISTS AND ANTAGONISTS AT MUSCARINIC RECEPTORS PRESENT ON ILEUM AND ATRIA INVITRO [J].
CLAGUE, RU ;
EGLEN, RM ;
STRACHAN, AC ;
WHITING, RL .
BRITISH JOURNAL OF PHARMACOLOGY, 1985, 86 (01) :163-170
[9]   INHIBITORY EFFECT OF GALLAMINE ON MUSCARINIC RECEPTORS [J].
CLARK, AL ;
MITCHELSON, F .
BRITISH JOURNAL OF PHARMACOLOGY, 1976, 58 (03) :323-331
[10]  
DEJONGE A, 1986, BRIT J PHARMACOL, V89, pP551