SYNTHESIS OF GEM-BISPHOSPHONIC CONJUGATES OF CORTISONE DERIVATIVES

被引：10

作者：

GUERVENOU, J

STURTZ, G

机构：

来源：

PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS | 1994年 / 88卷 / 1-4期

关键词：

GEM-BISPHOSPHONATE; GEM-BISPHOSPHONIC; TETRAETHYL ETHYLIDENE GEM-BISPHOSPHONATE; CORTICOSTEROIDS; ESTERIFICATION; ANTIINFLAMMATORY; DELIVERY-TARGETING CONCEPT;

D O I：

10.1080/10426509408036901

中图分类号：

O61 [无机化学];

学科分类号：

070301 ; 081704 ;

摘要：

Some gem-bisphosphonic cortico-steroid conjugates are prepared by esterification between gem-bisphosphonate carboxylic acids and steroid primary alcohols. These original products take place in a biological study about a delivery-targeting concept of active constituents in bone therapy, with the assistance of gem-bisphosphonic building-blocs.

引用

页码：1 / 13

页数：13

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