MULTIPLE CONFORMATIONAL STATES OF BENZODIAZEPINE RECEPTORS

被引:18
作者
CHIU, T
ROSENBERG, H
机构
关键词
D O I
10.1016/0165-6147(83)90435-2
中图分类号
R9 [药学];
学科分类号
1007 ;
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页码:348 / 350
页数:3
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[1]   [H-3]-LABELED PROPYL BETA-CARBOLINE-3-CARBOXYLATE AS A SELECTIVE RADIOLIGAND FOR THE BZ1 BENZODIAZEPINE RECEPTOR SUBCLASS [J].
BRAESTRUP, C ;
NIELSEN, M .
JOURNAL OF NEUROCHEMISTRY, 1981, 37 (02) :333-341
[2]  
CHIU TH, 1982, MOL PHARMACOL, V21, P57
[3]   COMPARISON OF THE KINETICS OF [H-3]-LABELED DIAZEPAM AND [H-3]-LABELED FLUNITRAZEPAM BINDING TO CORTICAL SYNAPTOSOMAL MEMBRANES [J].
CHIU, TH ;
ROSENBERG, HC .
JOURNAL OF NEUROCHEMISTRY, 1982, 39 (06) :1716-1725
[4]  
CHIU TH, MOL PHARM
[5]   REGIONAL HETEROGENEITY OF BENZODIAZEPINE RECEPTORS AT 37-DEGREES-C - AN INVITRO STUDY IN VARIOUS REGIONS OF THE RAT-BRAIN [J].
GEE, KW ;
YAMAMURA, HI .
LIFE SCIENCES, 1982, 31 (18) :1939-1945
[6]  
MACKERER CR, 1978, J PHARMACOL EXP THER, V206, P405
[7]   AGONIST AND ANTAGONIST BENZODIAZEPINE RECEPTOR INTERACTION INVITRO [J].
MOHLER, H ;
RICHARDS, JG .
NATURE, 1981, 294 (5843) :763-765
[8]   BENZODIAZEPINE RECEPTOR - DEMONSTRATION IN CENTRAL NERVOUS-SYSTEM [J].
MOHLER, H ;
OKADA, T .
SCIENCE, 1977, 198 (4319) :849-851
[9]   BENZODIAZEPINE RECEPTOR PROTEIN IDENTIFIED AND VISUALIZED IN BRAIN-TISSUE BY A PHOTOAFFINITY LABEL [J].
MOHLER, H ;
BATTERSBY, MK ;
RICHARDS, JG .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (03) :1666-1670
[10]   INTERACTION OF [H-3]-LABELED FLUNITRAZEPAM WITH THE BENZODIAZEPINE RECEPTOR - EVIDENCE FOR A LIGAND-INDUCED CONFORMATION CHANGE [J].
QUAST, U ;
MAHLMANN, H .
BIOCHEMICAL PHARMACOLOGY, 1982, 31 (17) :2761-2768