THE PERMEATION PATHWAY OF NEUROTRANSMITTER-GATED ION CHANNELS

被引:44
作者
LESTER, HA
机构
[1] Division of Biology, California Institute of Technology, Pasadena
来源
ANNUAL REVIEW OF BIOPHYSICS AND BIOMOLECULAR STRUCTURE | 1992年 / 21卷
关键词
SYNAPSE; NICOTINIC ACETYLCHOLINE RECEPTOR; NEUROTRANSMITTER RECEPTOR; OPEN-CHANNEL BLOCKERS; SITE-DIRECTED MUTAGENESIS;
D O I
10.1146/annurev.bb.21.060192.001411
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
[No abstract available]
引用
收藏
页码:267 / 292
页数:26
相关论文
共 161 条
[51]   A POSSIBLE MODEL FOR THE INNER WALL OF THE ACETYLCHOLINE-RECEPTOR CHANNEL [J].
FUROISCORBIN, S ;
PULLMAN, A .
BIOCHIMICA ET BIOPHYSICA ACTA, 1989, 984 (03) :339-350
[52]   ENERGY PROFILES IN THE ACETYLCHOLINE-RECEPTOR (ACHR) CHANNEL - THE MII-HELIX MODEL AND THE ROLE OF THE REMAINING HELICES [J].
FUROISCORBIN, S ;
PULLMAN, A .
FEBS LETTERS, 1989, 252 (1-2) :63-68
[53]   THE EFFECT OF POINT MUTATIONS ON ENERGY PROFILES IN A MODEL OF THE NICOTINIC ACETYLCHOLINE-RECEPTOR (ACHR) CHANNEL [J].
FUROISCORBIN, S ;
PULLMAN, A .
BIOPHYSICAL CHEMISTRY, 1991, 39 (02) :153-159
[54]   MINIATURE END-PLATE CURRENTS IN VOLTAGE-CLAMPED MUSCLE FIBRE [J].
GAGE, PW ;
ARMSTRONG, CM .
NATURE, 1968, 218 (5139) :363-+
[55]   FUNCTIONAL ARCHITECTURE OF THE NICOTINIC ACETYLCHOLINE-RECEPTOR - FROM ELECTRIC ORGAN TO BRAIN [J].
GALZI, JL ;
REVAH, F ;
BESSIS, A ;
CHANGEUX, JP .
ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, 1991, 31 :37-72
[56]   STRUCTURE OF THE HIGH-AFFINITY BINDING-SITE FOR NONCOMPETITIVE BLOCKERS OF THE ACETYLCHOLINE-RECEPTOR - SERINE-262 OF THE DELTA-SUBUNIT IS LABELED BY [H-3] CHLORPROMAZINE [J].
GIRAUDAT, J ;
DENNIS, M ;
HEIDMANN, T ;
CHANG, JY ;
CHANGEUX, JP .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1986, 83 (08) :2719-2723
[57]   STRUCTURE OF THE HIGH-AFFINITY BINDING-SITE FOR NONCOMPETITIVE BLOCKERS OF THE ACETYLCHOLINE-RECEPTOR - (H-3) CHLORPROMAZINE LABELS HOMOLOGOUS RESIDUES IN THE BETA-CHAIN AND DELTA-CHAIN [J].
GIRAUDAT, J ;
DENNIS, M ;
HEIDMANN, T ;
HAUMONT, PY ;
LEDERER, F ;
CHANGEUX, JP .
BIOCHEMISTRY, 1987, 26 (09) :2410-2418
[58]   THE CHANNEL-BLOCKING ACTION OF METHONIUM COMPOUNDS ON RAT SUBMANDIBULAR GANGLION-CELLS [J].
GURNEY, AM ;
RANG, HP .
BRITISH JOURNAL OF PHARMACOLOGY, 1984, 82 (03) :623-642
[59]   A STRUCTURAL MODEL OF THE ACETYLCHOLINE-RECEPTOR CHANNEL BASED ON PARTITION ENERGY AND HELIX PACKING CALCULATIONS [J].
GUY, HR .
BIOPHYSICAL JOURNAL, 1984, 45 (01) :249-261
[60]   THE ION CHANNEL OF THE NICOTINIC ACETYLCHOLINE-RECEPTOR [J].
GUY, HR ;
HUCHO, F .
TRENDS IN NEUROSCIENCES, 1987, 10 (08) :318-321