ADDITION OF DIAMINES TO METHYLTHIOPYRIDONES

被引:18
作者
HEHEMANN, DG
WINNIK, W
机构
[1] Department of Chemistry, Cleveland State University, Cleveland, Ohio
[2] NASA Lewis Research Center, Cleveland, Ohio, 44135, 21000 Brookpark Road
关键词
D O I
10.1002/jhet.5570310224
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
Thiopyridone derivatives react with diamines: ethylenediamine, 1,3-propylenediamine and 1,4-butylenediamine to produce bicyclic addition compounds. Ethanolamine reacts with thiopyridone derivatives to afford only open chain adducts. Diethylenetriamine and 2-(2-aminoethylamino)ethanol in reaction with thiopyridones yielded seven membered ring tricyclic derivatives. The procedures described here constitute a relatively simple method to prepare these novel heterocycles.
引用
收藏
页码:393 / 396
页数:4
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