RU-38486 - A POTENT ANTIGLUCOCORTICOID INVITRO AND INVIVO

被引:186
作者
GAGNE, D
PONS, M
PHILIBERT, D
机构
[1] INSERM,U58,60 RUE NAVACELLES,F-34100 MONTPELLIER,FRANCE
[2] CTR RECH ROUSSEL UCLAF,F-93230 ROMAINVILLE,FRANCE
关键词
D O I
10.1016/0022-4731(85)90401-7
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:247 / 251
页数:5
相关论文
共 31 条
  • [1] DNA-BINDING PROPERTIES OF GLUCOCORTICOSTEROID RECEPTORS BOUND TO THE STEROID ANTAGONIST RU-486
    BOURGEOIS, S
    PFAHL, M
    BAULIEU, EE
    [J]. EMBO JOURNAL, 1984, 3 (04) : 751 - 755
  • [2] AN APPROACH TO THE MECHANISM OF THE POTENT ANTIGLUCOCORTICOID - 17-BETA-HYDROXY-11-BETA-4-DIMETHYLAMINOPHENYL-17-ALPHA-PROPYNYL-ESTRA-4,9-DIEN-3-ONE
    CHASSEROTGOLAZ, S
    BECK, G
    [J]. JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1984, 21 (05) : 585 - 591
  • [3] ANTIGLUCOCORTICOID PROPERTIES OF RU-38486 IN A DIFFERENTIATED HEPATOMA-CELL LINE
    CHOBERT, MN
    BAROUKI, R
    FINIDORI, J
    AGGERBECK, M
    HANOUNE, J
    PHILIBERT, D
    DERAEDT, R
    [J]. BIOCHEMICAL PHARMACOLOGY, 1983, 32 (22) : 3481 - 3483
  • [4] DELTA-1,9(11)-11-DEOXYCORTISOL - AN IMPROVED GLUCOCORTICOID ANTAGONIST
    CHROUSOS, GP
    BARNES, KM
    SAUER, MA
    LORIAUX, DL
    CUTLER, GB
    [J]. ENDOCRINOLOGY, 1980, 107 (02) : 472 - 477
  • [5] DEVELOPMENT OF GLUCOCORTICOID ANTAGONISTS
    CHROUSOS, GP
    CUTLER, GB
    SAUER, M
    SIMONS, SS
    LORIAUX, DL
    [J]. PHARMACOLOGY & THERAPEUTICS, 1983, 20 (02) : 263 - 281
  • [6] CHROUSOS GP, STEROIDS, V40, P425
  • [7] CHROUSOS GP, 1982, PROGR RES CLIN APPLI, P152
  • [8] 11-DEOXYCORTISOL - GLUCOCORTICOID ANTAGONIST INVIVO
    CUTLER, GB
    BARNES, KM
    SAUER, MA
    LORIAUX, DL
    [J]. ENDOCRINOLOGY, 1979, 104 (06) : 1839 - 1844
  • [10] INVIVO STUDY OF THE ACTION OF ANTI-GLUCOCORTICOIDS ON THYMUS WEIGHT RATIO, ANTIBODY TITER AND THE ADRENAL-PITUITARY-HYPOTHALAMUS AXIS
    DUNCAN, MR
    DUNCAN, GR
    [J]. JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1979, 10 (03) : 245 - 259