SYNTHESIS OF ENANTIOMERICALLY PURE AMINO-ACIDS CONTAINING A 2-AMINO-4-THIAZOLYL SIDE-CHAIN

被引：8

作者：

PATT, WC

SKEEAN, RW

STEINBAUGH, BA

机构：

[1] Chemistry Department, Parke-Davis Pharmaceutical Research Division, Warner-Lambert Company, 2800 Plymouth Road Ann Arbor, Michigan

来源：

SYNTHETIC COMMUNICATIONS | 1990年 / 20卷 / 20期

关键词：

D O I：

10.1080/00397919008051532

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Enantiomerically pure 2-amino-4-thiazolyl containing amino acids were readily synthesized from commercially available derivatives of aspartic acid and glutamic acid, via reaction with diazomethane and further cyclization with thiourea. © 1990, Taylor & Francis Group, LLC. All rights reserved.

引用

页码：3097 / 3102

页数：6

共 8 条

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