CORRELATION ANALYSIS OF BAKERS STUDIES ON ENZYME INHIBITION .2. CHYMOTRYPSIN, TRYPSIN, THYMIDINE PHOSPHORYLASE, URIDINE PHOSPHORYLASE, THYMIDYLATE SYNTHETASE, CYTOSINE NUCLEOSIDE DEAMINASE, DIHYDROFOLATE-REDUCTASE, MALATE DEHYDROGENASE, GLUTAMATE-DEHYDROGENASE, LACTATE-DEHYDROGENASE, AND GLYCERALDEHYDE-PHOSPHATE DEHYDROGENASE

被引：60

作者：

YOSHIMOTO, M ^{[1
]}

HANSCH, C ^{[1
]}

机构：

[1] POMONA COLL,DEPT CHEM,CLAREMONT,CA 91711

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1976年 / 19卷 / 01期

关键词：

D O I：

10.1021/jm00223a015

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：71 / 98

页数：28

共 69 条

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[6] IRREVERSIBLE ENZYME INHIBITORS .104. INHIBITORS OF THYMIDINE PHOSPHORYLASE .8. FURTHER STUDIES ON HYDROPHOBIC BONDING WITH 6-SUBSTITUTED URACILS [J].

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[7] ANALOGS OF TETRAHYDROFOLIC ACID .24. FURTHER OBSERVATIONS ON MODE OF PYRIMIDYL BINDING TO DIHYDROFOLIC REDUCTASE AND THYMIDYLATE SYNTHETASE BY 2-AMINO-5-(3-ANILINOPROPYL)-6-METHYL-4-PYRIMIDINOL TYPE OF INHIBITOR [J].

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[10] ANALOGS OF TETRAHYDROFOLIC ACID .27. HYDROPHOBIC BONDING TO DIHYDROFOLIC REDUCTASE BY 2-AMINO-4,6-DISUBSTITUTED-5-ALKYLPYRIMIDINES AND 1-ALKYL-4,6-DIAMINO-1,2-DIHYDRO-S-TRIAZINES [J].

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