SYNTHESIS AND INVIVO STUDIES OF THE RADIOSENSITIZER 4-[BR-82]BROMOMISONIDAZOLE

被引:40
作者
JETTE, DC [1 ]
WIEBE, LI [1 ]
CHAPMAN, JD [1 ]
机构
[1] UNIV ALBERTA,FAC PHARM & PHARMACEUT SCI,EDMONTON T6G 2N8,ALBERTA,CANADA
来源
INTERNATIONAL JOURNAL OF NUCLEAR MEDICINE & BIOLOGY | 1983年 / 10卷 / 04期
关键词
D O I
10.1016/0047-0740(83)90080-3
中图分类号
R8 [特种医学]; R445 [影像诊断学];
学科分类号
1002 ; 100207 ; 1009 ;
摘要
引用
收藏
页码:205 / 210
页数:6
相关论文
共 15 条
[1]   DISTRIBUTION OF MISONIDAZOLE IN HUMAN-TUMORS AND NORMAL-TISSUES [J].
ASH, DV ;
SMITH, MR ;
BUGDEN, RD .
BRITISH JOURNAL OF CANCER, 1979, 39 (05) :503-509
[2]   PHARMACOKINETIC CONSIDERATIONS IN TESTING HYPOXIC CELL RADIOSENSITIZERS IN MOUSE-TUMORS [J].
BROWN, JM ;
YU, NY ;
WORKMAN, P .
BRITISH JOURNAL OF CANCER, 1979, 39 (03) :310-320
[3]   A MARKER FOR HYPOXIC CELLS IN TUMORS WITH POTENTIAL CLINICAL APPLICABILITY [J].
CHAPMAN, JD ;
FRANKO, AJ ;
SHARPLIN, J .
BRITISH JOURNAL OF CANCER, 1981, 43 (04) :546-550
[4]   THE METABOLISM AND PHARMACOKINETICS OF THE HYPOXIC CELL RADIOSENSITIZER AND CYTO-TOXIC AGENT, MISONIDAZOLE, IN C3H MICE [J].
CHIN, JB ;
RAUTH, AM .
RADIATION RESEARCH, 1981, 86 (02) :341-357
[5]   CLINICAL TESTING OF RADIOSENSITIZER RO 07-0582 - EXPERIENCE WITH MULTIPLE DOSES [J].
DISCHE, S ;
SAUNDERS, MI ;
LEE, ME ;
ADAMS, GE ;
FLOCKHART, IR .
BRITISH JOURNAL OF CANCER, 1977, 35 (05) :567-579
[6]  
GARRECHT B, BR J CANCER
[7]  
JETTE DC, 1981, UASF ANN REP R, V20
[8]   TUMOR UPTAKE OF RADIOLABELED PYRIMIDINE-BASES AND PYRIMIDINE NUCLEOSIDES IN ANIMAL-MODELS .3. 2'-[BR-82]-BROMO-2'-DEOXYURIDINE [J].
LEE, YW ;
KNAUS, EE ;
WIEBE, LI .
INTERNATIONAL JOURNAL OF NUCLEAR MEDICINE & BIOLOGY, 1979, 6 (02) :109-112
[9]   DISTRIBUTION AND TUMOR-CYTOTOXICITY OF THE RADIOSENSITIZER MISONIDAZOLE (RO-07-0582) IN C57 MICE [J].
PEDERSEN, JE ;
SMITH, MR ;
BUGDEN, RD ;
PECKHAM, MJ .
BRITISH JOURNAL OF CANCER, 1979, 39 (04) :429-433
[10]  
SOREMARK R, 1960, ACTA RADIOL S, V190, P23