THE POLYMORPHIC OXIDATION OF BETA-ADRENOCEPTOR ANTAGONISTS - CLINICAL PHARMACOKINETIC CONSIDERATIONS

被引:82
作者
LENNARD, MS
TUCKER, GT
WOODS, HF
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关键词
D O I
10.2165/00003088-198611010-00001
中图分类号
R9 [药学];
学科分类号
1007 ;
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页码:1 / 17
页数:17
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共 93 条
[1]  
ALVAN G, 1982, LANCET, V1, P333
[2]   METABOLISM OF METOPROLOL IN RAT INVITRO AND INVIVO [J].
ARFWIDSSON, A ;
BORG, KO ;
HOFFMANN, KJ ;
SKANBERG, I .
XENOBIOTICA, 1976, 6 (11) :691-711
[3]  
BAI SA, 1983, J PHARMACOL EXP THER, V224, P62
[4]  
BAI TR, 1982, J ROY COLL PHYS LOND, V16, P239
[5]   INFLUENCE OF RENAL-FAILURE ON THE HEPATIC-CLEARANCE OF BUFURALOL IN MAN [J].
BALANT, L ;
FRANCIS, RJ ;
TOZER, TN ;
MARMY, A ;
TSCHOPP, JM ;
FABRE, J .
JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1980, 8 (05) :421-438
[6]  
BALANT L, 1976, SCHWEIZ MED WSCHR, V106, P1403
[7]   INHIBITION OF ANTIPYRINE METABOLISM BY BETA-ADRENOCEPTOR ANTAGONISTS [J].
BAX, NDS ;
LENNARD, MS ;
TUCKER, GT .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1981, 12 (06) :779-784
[8]   PHARMACOGENETIC COVARIATION OF DEFECTIVE N-OXIDATION OF SPARTEINE AND 4-HYDROXYLATION OF DEBRISOQUINE [J].
BERTILSSON, L ;
DENGLER, HJ ;
EICHELBAUM, M ;
SCHULZ, HU .
EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1980, 17 (02) :153-155
[9]  
BOOBIS AR, 1983, MOL PHARMACOL, V23, P474
[10]   GENETIC-POLYMORPHISM IN DRUG OXIDATION - INVITRO STUDIES OF HUMAN DEBRISOQUINE 4-HYDROXYLASE AND BUFURALOL 1'-HYDROXYLASE ACTIVITIES [J].
BOOBIS, AR ;
MURRAY, S ;
HAMPDEN, CE ;
DAVIES, DS .
BIOCHEMICAL PHARMACOLOGY, 1985, 34 (01) :65-71