THE POLYMORPHIC OXIDATION OF BETA-ADRENOCEPTOR ANTAGONISTS - CLINICAL PHARMACOKINETIC CONSIDERATIONS

被引:82
作者
LENNARD, MS
TUCKER, GT
WOODS, HF
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关键词
D O I
10.2165/00003088-198611010-00001
中图分类号
R9 [药学];
学科分类号
1007 ;
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页码:1 / 17
页数:17
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共 93 条
[61]  
LENNARD MS, 1985, XENOBIOTICA
[62]  
LENNARD MS, 1983, PHARM INT, V4, P61
[63]   TIMOLOL AND ATENOLOL - RELATIONSHIPS BETWEEN OXIDATION PHENOTYPE, PHARMACOKINETICS AND PHARMACODYNAMICS [J].
LEWIS, RV ;
LENNARD, MS ;
JACKSON, PR ;
TUCKER, GT ;
RAMSAY, LE ;
WOODS, HF .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1985, 19 (03) :329-333
[64]  
LOHMOLLER G, 1982, Z KARDIOL, V71, P619
[65]   POLYMORPHIC HYDROXYLATION OF DEBRISOQUINE IN MAN [J].
MAHGOUB, A ;
IDLE, JR ;
DRING, LG ;
LANCASTER, R ;
SMITH, RL .
LANCET, 1977, 2 (8038) :584-586
[66]   A STUDY OF THE DEBRISOQUINE HYDROXYLATION POLYMORPHISM IN A NIGERIAN POPULATION [J].
MBANEFO, C ;
BABABUNMI, EA ;
MAHGOUB, A ;
SLOAN, TP ;
IDLE, JR ;
SMITH, RL .
XENOBIOTICA, 1980, 10 (11) :811-818
[67]   PHARMACOKINETICS AND BETA-BLOCKING EFFECTS OF TIMOLOL IN POOR AND EXTENSIVE METABOLIZERS OF DEBRISOQUIN [J].
MCGOURTY, JC ;
SILAS, JH ;
FLEMING, JJ ;
MCBURNEY, A ;
WARD, JW .
CLINICAL PHARMACOLOGY & THERAPEUTICS, 1985, 38 (04) :409-413
[68]   METOPROLOL METABOLISM AND DEBRISOQUINE OXIDATION POLYMORPHISM - POPULATION AND FAMILY STUDIES [J].
MCGOURTY, JC ;
SILAS, JH ;
LENNARD, MS ;
TUCKER, GT ;
WOODS, HF .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1985, 20 (06) :555-566
[69]  
MEIER PJ, 1983, GASTROENTEROLOGY, V85, P682
[70]   BUFURALOL METABOLISM IN HUMAN-LIVER - A SENSITIVE PROBE FOR THE DEBRISOQUINE-TYPE POLYMORPHISM OF DRUG OXIDATION [J].
MINDER, EI ;
MEIER, PJ ;
MULLER, HK ;
MINDER, C ;
MEYER, UA .
EUROPEAN JOURNAL OF CLINICAL INVESTIGATION, 1984, 14 (03) :184-189