K-252A, A POTENT INHIBITOR OF PROTEIN-KINASE-C FROM MICROBIAL ORIGIN

被引:349
作者
KASE, H
IWAHASHI, K
MATSUDA, Y
机构
关键词
D O I
10.7164/antibiotics.39.1059
中图分类号
Q81 [生物工程学(生物技术)]; Q93 [微生物学];
学科分类号
071005 ; 0836 ; 090102 ; 100705 ;
摘要
引用
收藏
页码:1059 / 1065
页数:7
相关论文
共 25 条
[1]  
Ames BN, 1966, METHOD ENZYMOL, V8, P115, DOI DOI 10.1016/0076-6879(66)08014-5
[2]  
BRADFORD MM, 1976, ANAL BIOCHEM, V72, P248, DOI 10.1016/0003-2697(76)90527-3
[3]  
BUTCHER RW, 1962, J BIOL CHEM, V237, P1244
[5]   CALMODULIN PLAYS A PIVOTAL ROLE IN CELLULAR-REGULATION [J].
CHEUNG, WY .
SCIENCE, 1980, 207 (4426) :19-27
[6]   ISOQUINOLINESULFONAMIDES, NOVEL AND POTENT INHIBITORS OF CYCLIC-NUCLEOTIDE DEPENDENT PROTEIN-KINASE AND PROTEIN KINASE-C [J].
HIDAKA, H ;
INAGAKI, M ;
KAWAMOTO, S ;
SASAKI, Y .
BIOCHEMISTRY, 1984, 23 (21) :5036-5041
[8]   MULTIPLE CYCLIC NUCLEOTIDE PHOSPHODIESTERASE ACTIVITIES FROM RAT TISSUES AND OCCURRENCE OF A CALCIUM-PLUS-MAGNESIUM-ION-DEPENDENT PHOSPHODIESTERASE AND ITS PROTEIN ACTIVATOR [J].
KAKIUCHI, S ;
YAMAZAKI, R ;
TESHIMA, Y ;
UENISHI, K ;
MIYAMOTO, E .
BIOCHEMICAL JOURNAL, 1975, 146 (01) :109-120
[9]  
KIKKAWA U, 1982, J BIOL CHEM, V257, P13341
[10]   A NEW ANTIBIOTIC SF-2370 PRODUCED BY ACTINOMADURA [J].
KOYAMA, M ;
KAI, F ;
SHOMURA, T ;
KOJIMA, M .
JOURNAL OF ANTIBIOTICS, 1985, 38 (10) :1437-1439