K-252A, A POTENT INHIBITOR OF PROTEIN-KINASE-C FROM MICROBIAL ORIGIN

被引:349
作者
KASE, H
IWAHASHI, K
MATSUDA, Y
机构
关键词
D O I
10.7164/antibiotics.39.1059
中图分类号
Q81 [生物工程学(生物技术)]; Q93 [微生物学];
学科分类号
071005 ; 0836 ; 090102 ; 100705 ;
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页码:1059 / 1065
页数:7
相关论文
共 25 条
[21]  
TANAKA T, 1982, MOL PHARMACOL, V22, P408
[22]   BASIC-PROTEIN IN BRAIN MYELIN IS PHOSPHORYLATED BY ENDOGENOUS PHOSPHOLIPID-SENSITIVE CA-2+-DEPENDENT PROTEIN-KINASE [J].
TURNER, RS ;
CHOU, CHJ ;
KIBLER, RF ;
KUO, JF .
JOURNAL OF NEUROCHEMISTRY, 1982, 39 (05) :1397-1404
[23]   INHIBITION BY PHENOTHIAZINE ANTIPSYCHOTIC-DRUGS OF CALCIUM-DEPENDENT PHOSPHORYLATION OF CEREBRAL-CORTEX PROTEINS REGULATED BY PHOSPHOLIPID OR CALMODULIN [J].
WRENN, RW ;
KATOH, N ;
SCHATZMAN, RC ;
KUO, JF .
LIFE SCIENCES, 1981, 29 (07) :725-733
[24]  
YAMADA K, 1986, JPN J PHARMACOL, V40, pP265
[25]   THE STRUCTURES OF THE NOVEL PROTEIN-KINASE-C INHIBITORS K-252A, B, C AND D [J].
YASUZAWA, T ;
IIDA, T ;
YOSHIDA, M ;
HIRAYAMA, N ;
TAKAHASHI, M ;
SHIRAHATA, K ;
SANO, H .
JOURNAL OF ANTIBIOTICS, 1986, 39 (08) :1072-1078