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A-69024 - A NON-BENZAZEPINE ANTAGONIST WITH SELECTIVITY FOR THE DOPAMINE D-1 RECEPTOR
被引:38
作者
:
KERKMAN, DJ
论文数:
0
引用数:
0
h-index:
0
KERKMAN, DJ
ACKERMAN, M
论文数:
0
引用数:
0
h-index:
0
ACKERMAN, M
ARTMAN, LD
论文数:
0
引用数:
0
h-index:
0
ARTMAN, LD
MACKENZIE, RG
论文数:
0
引用数:
0
h-index:
0
MACKENZIE, RG
JOHNSON, MC
论文数:
0
引用数:
0
h-index:
0
JOHNSON, MC
BEDNARZ, L
论文数:
0
引用数:
0
h-index:
0
BEDNARZ, L
MONTANA, W
论文数:
0
引用数:
0
h-index:
0
MONTANA, W
ASIN, KE
论文数:
0
引用数:
0
h-index:
0
ASIN, KE
STAMPFLI, H
论文数:
0
引用数:
0
h-index:
0
STAMPFLI, H
KEBABIAN, JW
论文数:
0
引用数:
0
h-index:
0
KEBABIAN, JW
机构
:
来源
:
EUROPEAN JOURNAL OF PHARMACOLOGY
|
1989年
/ 166卷
/ 03期
关键词
:
D O I
:
10.1016/0014-2999(89)90362-2
中图分类号
:
R9 [药学];
学科分类号
:
1007 ;
摘要
:
引用
收藏
页码:481 / 491
页数:11
相关论文
共 33 条
[1]
EVIDENCE FOR DIFFERENT STATES OF THE DOPAMINE D1 RECEPTOR - CLOZAPINE AND FLUPERLAPINE MAY PREFERENTIALLY LABEL AN ADENYLATE CYCLASE-COUPLED STATE OF THE D1-RECEPTOR
ANDERSEN, PH
论文数:
0
引用数:
0
h-index:
0
机构:
ST HANS MENTAL HOSP, PSYCHOPHARMACOL RES LAB, DK-4000 ROSKILDE, DENMARK
ST HANS MENTAL HOSP, PSYCHOPHARMACOL RES LAB, DK-4000 ROSKILDE, DENMARK
ANDERSEN, PH
BRAESTRUP, C
论文数:
0
引用数:
0
h-index:
0
机构:
ST HANS MENTAL HOSP, PSYCHOPHARMACOL RES LAB, DK-4000 ROSKILDE, DENMARK
ST HANS MENTAL HOSP, PSYCHOPHARMACOL RES LAB, DK-4000 ROSKILDE, DENMARK
BRAESTRUP, C
[J].
JOURNAL OF NEUROCHEMISTRY,
1986,
47
(06)
: 1822
-
1831
[2]
SOME ATYPICAL NEUROLEPTICS INHIBIT [H-3] SCH 23390 BINDING INVIVO
ANDERSEN, PH
论文数:
0
引用数:
0
h-index:
0
机构:
NOVO PHARMACEUT RES & DEV,DEPT MED CHEM 1,DK-2880 BAGSVAERD,DENMARK
NOVO PHARMACEUT RES & DEV,DEPT MED CHEM 1,DK-2880 BAGSVAERD,DENMARK
ANDERSEN, PH
NIELSEN, EB
论文数:
0
引用数:
0
h-index:
0
机构:
NOVO PHARMACEUT RES & DEV,DEPT MED CHEM 1,DK-2880 BAGSVAERD,DENMARK
NOVO PHARMACEUT RES & DEV,DEPT MED CHEM 1,DK-2880 BAGSVAERD,DENMARK
NIELSEN, EB
GRONVALD, FC
论文数:
0
引用数:
0
h-index:
0
机构:
NOVO PHARMACEUT RES & DEV,DEPT MED CHEM 1,DK-2880 BAGSVAERD,DENMARK
NOVO PHARMACEUT RES & DEV,DEPT MED CHEM 1,DK-2880 BAGSVAERD,DENMARK
GRONVALD, FC
BRAESTRUP, C
论文数:
0
引用数:
0
h-index:
0
机构:
NOVO PHARMACEUT RES & DEV,DEPT MED CHEM 1,DK-2880 BAGSVAERD,DENMARK
NOVO PHARMACEUT RES & DEV,DEPT MED CHEM 1,DK-2880 BAGSVAERD,DENMARK
BRAESTRUP, C
[J].
EUROPEAN JOURNAL OF PHARMACOLOGY,
1986,
120
(01)
: 143
-
144
[3]
DIFFERENTIAL INVOLVEMENT OF DOPAMINE D-1 AND D-2 RECEPTORS IN THE CIRCLING BEHAVIOR INDUCED BY APOMORPHINE, SK+F-38393, PERGOLIDE AND LY-171555 IN 6-HYDROXYDOPAMINE-LESIONED RATS
ARNT, J
论文数:
0
引用数:
0
h-index:
0
ARNT, J
HYTTEL, J
论文数:
0
引用数:
0
h-index:
0
HYTTEL, J
[J].
PSYCHOPHARMACOLOGY,
1985,
85
(03)
: 346
-
352
[4]
SYNTHESIS AND PHARMACOLOGICAL CHARACTERIZATION OF 1-PHENYL-1,2,3,4-TETRAHYDROISOQUINOLINE, 4-PHENYL-1,2,3,4-TETRAHYDROISOQUINOLINE, AND 1-BENZYL-1,2,3,4-TETRAHYDROISOQUINOLINE AS DOPAMINE RECEPTOR LIGANDS
CHARIFSON, PS
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV N CAROLINA,SCH PHARM,DIV MED CHEM & NAT PROD,CHAPEL HILL,NC 27599
CHARIFSON, PS
WYRICK, SD
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV N CAROLINA,SCH PHARM,DIV MED CHEM & NAT PROD,CHAPEL HILL,NC 27599
WYRICK, SD
HOFFMAN, AJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV N CAROLINA,SCH PHARM,DIV MED CHEM & NAT PROD,CHAPEL HILL,NC 27599
HOFFMAN, AJ
SIMMONS, RMA
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV N CAROLINA,SCH PHARM,DIV MED CHEM & NAT PROD,CHAPEL HILL,NC 27599
SIMMONS, RMA
BOWEN, JP
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV N CAROLINA,SCH PHARM,DIV MED CHEM & NAT PROD,CHAPEL HILL,NC 27599
BOWEN, JP
MCDOUGALD, DL
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV N CAROLINA,SCH PHARM,DIV MED CHEM & NAT PROD,CHAPEL HILL,NC 27599
MCDOUGALD, DL
MAILMAN, RB
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV N CAROLINA,SCH PHARM,DIV MED CHEM & NAT PROD,CHAPEL HILL,NC 27599
MAILMAN, RB
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1988,
31
(10)
: 1941
-
1946
[5]
CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099
[6]
PHARMACOLOGICAL EFFECTS OF A SPECIFIC DOPAMINE D-1 ANTAGONIST SCH-23390 IN COMPARISON WITH NEUROLEPTICS
CHRISTENSEN, AV
论文数:
0
引用数:
0
h-index:
0
CHRISTENSEN, AV
ARNT, J
论文数:
0
引用数:
0
h-index:
0
ARNT, J
HYTTEL, J
论文数:
0
引用数:
0
h-index:
0
HYTTEL, J
LARSEN, JJ
论文数:
0
引用数:
0
h-index:
0
LARSEN, JJ
SVENDSEN, O
论文数:
0
引用数:
0
h-index:
0
SVENDSEN, O
[J].
LIFE SCIENCES,
1984,
34
(16)
: 1529
-
1540
[7]
REVIEW - D1 DOPAMINE RECEPTOR - THE SEARCH FOR A FUNCTION - A CRITICAL-EVALUATION OF THE D1/D2 DOPAMINE RECEPTOR CLASSIFICATION AND ITS FUNCTIONAL IMPLICATIONS
CLARK, D
论文数:
0
引用数:
0
h-index:
0
机构:
SINAI HOSP, CTR CELL BIOL, NEUROPHYSIOL LAB, DETROIT, MI 48235 USA
CLARK, D
WHITE, FJ
论文数:
0
引用数:
0
h-index:
0
机构:
SINAI HOSP, CTR CELL BIOL, NEUROPHYSIOL LAB, DETROIT, MI 48235 USA
WHITE, FJ
[J].
SYNAPSE,
1987,
1
(04)
: 347
-
388
[8]
D-2 DOPAMINE RECEPTOR-MEDIATED INHIBITION OF ADENYLATE-CYCLASE ACTIVITY IN THE INTERMEDIATE LOBE OF THE RAT PITUITARY-GLAND REQUIRES GUANOSINE 5'-TRIPHOSPHATE
COTE, TE
论文数:
0
引用数:
0
h-index:
0
机构:
NINCDS,EXPTL THERAPEUT BRANCH,BETHESDA,MD 20205
NINCDS,EXPTL THERAPEUT BRANCH,BETHESDA,MD 20205
COTE, TE
GREWE, CW
论文数:
0
引用数:
0
h-index:
0
机构:
NINCDS,EXPTL THERAPEUT BRANCH,BETHESDA,MD 20205
NINCDS,EXPTL THERAPEUT BRANCH,BETHESDA,MD 20205
GREWE, CW
TSURUTA, K
论文数:
0
引用数:
0
h-index:
0
机构:
NINCDS,EXPTL THERAPEUT BRANCH,BETHESDA,MD 20205
NINCDS,EXPTL THERAPEUT BRANCH,BETHESDA,MD 20205
TSURUTA, K
STOOF, JC
论文数:
0
引用数:
0
h-index:
0
机构:
NINCDS,EXPTL THERAPEUT BRANCH,BETHESDA,MD 20205
NINCDS,EXPTL THERAPEUT BRANCH,BETHESDA,MD 20205
STOOF, JC
ESKAY, RL
论文数:
0
引用数:
0
h-index:
0
机构:
NINCDS,EXPTL THERAPEUT BRANCH,BETHESDA,MD 20205
NINCDS,EXPTL THERAPEUT BRANCH,BETHESDA,MD 20205
ESKAY, RL
KEBABIAN, JW
论文数:
0
引用数:
0
h-index:
0
机构:
NINCDS,EXPTL THERAPEUT BRANCH,BETHESDA,MD 20205
NINCDS,EXPTL THERAPEUT BRANCH,BETHESDA,MD 20205
KEBABIAN, JW
[J].
ENDOCRINOLOGY,
1982,
110
(03)
: 812
-
819
[9]
DOPAMINE-DERIVED ALKALOIDS IN ALCOHOLISM AND IN PARKINSONS AND HUNTINGTONS DISEASES
DOSTERT, P
论文数:
0
引用数:
0
h-index:
0
机构:
CHU CLERMONT FERRAND,F-63003 CLERMONT FERRAND,FRANCE
CHU CLERMONT FERRAND,F-63003 CLERMONT FERRAND,FRANCE
DOSTERT, P
BENEDETTI, MS
论文数:
0
引用数:
0
h-index:
0
机构:
CHU CLERMONT FERRAND,F-63003 CLERMONT FERRAND,FRANCE
CHU CLERMONT FERRAND,F-63003 CLERMONT FERRAND,FRANCE
BENEDETTI, MS
DORDAIN, G
论文数:
0
引用数:
0
h-index:
0
机构:
CHU CLERMONT FERRAND,F-63003 CLERMONT FERRAND,FRANCE
CHU CLERMONT FERRAND,F-63003 CLERMONT FERRAND,FRANCE
DORDAIN, G
[J].
JOURNAL OF NEURAL TRANSMISSION,
1988,
74
(02)
: 61
-
74
[10]
REGULATION OF AGONIST AND ANTAGONIST BINDING TO STRIATAL D-1 DOPAMINE-RECEPTORS - STUDIES USING THE SELECTIVE D-1 ANTAGONIST [H-3] SK-AND-F R-83566
FLAIM, KE
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS, DEPT RADIOCHEM, SWEDELAND, PA 19479 USA
FLAIM, KE
GESSNER, GW
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS, DEPT RADIOCHEM, SWEDELAND, PA 19479 USA
GESSNER, GW
CROOKE, ST
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS, DEPT RADIOCHEM, SWEDELAND, PA 19479 USA
CROOKE, ST
HEYS, JR
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS, DEPT RADIOCHEM, SWEDELAND, PA 19479 USA
HEYS, JR
WEINSTOCK, J
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS, DEPT RADIOCHEM, SWEDELAND, PA 19479 USA
WEINSTOCK, J
[J].
LIFE SCIENCES,
1986,
38
(23)
: 2087
-
2096
←
1
2
3
4
→
共 33 条
[1]
EVIDENCE FOR DIFFERENT STATES OF THE DOPAMINE D1 RECEPTOR - CLOZAPINE AND FLUPERLAPINE MAY PREFERENTIALLY LABEL AN ADENYLATE CYCLASE-COUPLED STATE OF THE D1-RECEPTOR
ANDERSEN, PH
论文数:
0
引用数:
0
h-index:
0
机构:
ST HANS MENTAL HOSP, PSYCHOPHARMACOL RES LAB, DK-4000 ROSKILDE, DENMARK
ST HANS MENTAL HOSP, PSYCHOPHARMACOL RES LAB, DK-4000 ROSKILDE, DENMARK
ANDERSEN, PH
BRAESTRUP, C
论文数:
0
引用数:
0
h-index:
0
机构:
ST HANS MENTAL HOSP, PSYCHOPHARMACOL RES LAB, DK-4000 ROSKILDE, DENMARK
ST HANS MENTAL HOSP, PSYCHOPHARMACOL RES LAB, DK-4000 ROSKILDE, DENMARK
BRAESTRUP, C
[J].
JOURNAL OF NEUROCHEMISTRY,
1986,
47
(06)
: 1822
-
1831
[2]
SOME ATYPICAL NEUROLEPTICS INHIBIT [H-3] SCH 23390 BINDING INVIVO
ANDERSEN, PH
论文数:
0
引用数:
0
h-index:
0
机构:
NOVO PHARMACEUT RES & DEV,DEPT MED CHEM 1,DK-2880 BAGSVAERD,DENMARK
NOVO PHARMACEUT RES & DEV,DEPT MED CHEM 1,DK-2880 BAGSVAERD,DENMARK
ANDERSEN, PH
NIELSEN, EB
论文数:
0
引用数:
0
h-index:
0
机构:
NOVO PHARMACEUT RES & DEV,DEPT MED CHEM 1,DK-2880 BAGSVAERD,DENMARK
NOVO PHARMACEUT RES & DEV,DEPT MED CHEM 1,DK-2880 BAGSVAERD,DENMARK
NIELSEN, EB
GRONVALD, FC
论文数:
0
引用数:
0
h-index:
0
机构:
NOVO PHARMACEUT RES & DEV,DEPT MED CHEM 1,DK-2880 BAGSVAERD,DENMARK
NOVO PHARMACEUT RES & DEV,DEPT MED CHEM 1,DK-2880 BAGSVAERD,DENMARK
GRONVALD, FC
BRAESTRUP, C
论文数:
0
引用数:
0
h-index:
0
机构:
NOVO PHARMACEUT RES & DEV,DEPT MED CHEM 1,DK-2880 BAGSVAERD,DENMARK
NOVO PHARMACEUT RES & DEV,DEPT MED CHEM 1,DK-2880 BAGSVAERD,DENMARK
BRAESTRUP, C
[J].
EUROPEAN JOURNAL OF PHARMACOLOGY,
1986,
120
(01)
: 143
-
144
[3]
DIFFERENTIAL INVOLVEMENT OF DOPAMINE D-1 AND D-2 RECEPTORS IN THE CIRCLING BEHAVIOR INDUCED BY APOMORPHINE, SK+F-38393, PERGOLIDE AND LY-171555 IN 6-HYDROXYDOPAMINE-LESIONED RATS
ARNT, J
论文数:
0
引用数:
0
h-index:
0
ARNT, J
HYTTEL, J
论文数:
0
引用数:
0
h-index:
0
HYTTEL, J
[J].
PSYCHOPHARMACOLOGY,
1985,
85
(03)
: 346
-
352
[4]
SYNTHESIS AND PHARMACOLOGICAL CHARACTERIZATION OF 1-PHENYL-1,2,3,4-TETRAHYDROISOQUINOLINE, 4-PHENYL-1,2,3,4-TETRAHYDROISOQUINOLINE, AND 1-BENZYL-1,2,3,4-TETRAHYDROISOQUINOLINE AS DOPAMINE RECEPTOR LIGANDS
CHARIFSON, PS
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV N CAROLINA,SCH PHARM,DIV MED CHEM & NAT PROD,CHAPEL HILL,NC 27599
CHARIFSON, PS
WYRICK, SD
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV N CAROLINA,SCH PHARM,DIV MED CHEM & NAT PROD,CHAPEL HILL,NC 27599
WYRICK, SD
HOFFMAN, AJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV N CAROLINA,SCH PHARM,DIV MED CHEM & NAT PROD,CHAPEL HILL,NC 27599
HOFFMAN, AJ
SIMMONS, RMA
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV N CAROLINA,SCH PHARM,DIV MED CHEM & NAT PROD,CHAPEL HILL,NC 27599
SIMMONS, RMA
BOWEN, JP
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV N CAROLINA,SCH PHARM,DIV MED CHEM & NAT PROD,CHAPEL HILL,NC 27599
BOWEN, JP
MCDOUGALD, DL
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV N CAROLINA,SCH PHARM,DIV MED CHEM & NAT PROD,CHAPEL HILL,NC 27599
MCDOUGALD, DL
MAILMAN, RB
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV N CAROLINA,SCH PHARM,DIV MED CHEM & NAT PROD,CHAPEL HILL,NC 27599
MAILMAN, RB
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1988,
31
(10)
: 1941
-
1946
[5]
CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099
[6]
PHARMACOLOGICAL EFFECTS OF A SPECIFIC DOPAMINE D-1 ANTAGONIST SCH-23390 IN COMPARISON WITH NEUROLEPTICS
CHRISTENSEN, AV
论文数:
0
引用数:
0
h-index:
0
CHRISTENSEN, AV
ARNT, J
论文数:
0
引用数:
0
h-index:
0
ARNT, J
HYTTEL, J
论文数:
0
引用数:
0
h-index:
0
HYTTEL, J
LARSEN, JJ
论文数:
0
引用数:
0
h-index:
0
LARSEN, JJ
SVENDSEN, O
论文数:
0
引用数:
0
h-index:
0
SVENDSEN, O
[J].
LIFE SCIENCES,
1984,
34
(16)
: 1529
-
1540
[7]
REVIEW - D1 DOPAMINE RECEPTOR - THE SEARCH FOR A FUNCTION - A CRITICAL-EVALUATION OF THE D1/D2 DOPAMINE RECEPTOR CLASSIFICATION AND ITS FUNCTIONAL IMPLICATIONS
CLARK, D
论文数:
0
引用数:
0
h-index:
0
机构:
SINAI HOSP, CTR CELL BIOL, NEUROPHYSIOL LAB, DETROIT, MI 48235 USA
CLARK, D
WHITE, FJ
论文数:
0
引用数:
0
h-index:
0
机构:
SINAI HOSP, CTR CELL BIOL, NEUROPHYSIOL LAB, DETROIT, MI 48235 USA
WHITE, FJ
[J].
SYNAPSE,
1987,
1
(04)
: 347
-
388
[8]
D-2 DOPAMINE RECEPTOR-MEDIATED INHIBITION OF ADENYLATE-CYCLASE ACTIVITY IN THE INTERMEDIATE LOBE OF THE RAT PITUITARY-GLAND REQUIRES GUANOSINE 5'-TRIPHOSPHATE
COTE, TE
论文数:
0
引用数:
0
h-index:
0
机构:
NINCDS,EXPTL THERAPEUT BRANCH,BETHESDA,MD 20205
NINCDS,EXPTL THERAPEUT BRANCH,BETHESDA,MD 20205
COTE, TE
GREWE, CW
论文数:
0
引用数:
0
h-index:
0
机构:
NINCDS,EXPTL THERAPEUT BRANCH,BETHESDA,MD 20205
NINCDS,EXPTL THERAPEUT BRANCH,BETHESDA,MD 20205
GREWE, CW
TSURUTA, K
论文数:
0
引用数:
0
h-index:
0
机构:
NINCDS,EXPTL THERAPEUT BRANCH,BETHESDA,MD 20205
NINCDS,EXPTL THERAPEUT BRANCH,BETHESDA,MD 20205
TSURUTA, K
STOOF, JC
论文数:
0
引用数:
0
h-index:
0
机构:
NINCDS,EXPTL THERAPEUT BRANCH,BETHESDA,MD 20205
NINCDS,EXPTL THERAPEUT BRANCH,BETHESDA,MD 20205
STOOF, JC
ESKAY, RL
论文数:
0
引用数:
0
h-index:
0
机构:
NINCDS,EXPTL THERAPEUT BRANCH,BETHESDA,MD 20205
NINCDS,EXPTL THERAPEUT BRANCH,BETHESDA,MD 20205
ESKAY, RL
KEBABIAN, JW
论文数:
0
引用数:
0
h-index:
0
机构:
NINCDS,EXPTL THERAPEUT BRANCH,BETHESDA,MD 20205
NINCDS,EXPTL THERAPEUT BRANCH,BETHESDA,MD 20205
KEBABIAN, JW
[J].
ENDOCRINOLOGY,
1982,
110
(03)
: 812
-
819
[9]
DOPAMINE-DERIVED ALKALOIDS IN ALCOHOLISM AND IN PARKINSONS AND HUNTINGTONS DISEASES
DOSTERT, P
论文数:
0
引用数:
0
h-index:
0
机构:
CHU CLERMONT FERRAND,F-63003 CLERMONT FERRAND,FRANCE
CHU CLERMONT FERRAND,F-63003 CLERMONT FERRAND,FRANCE
DOSTERT, P
BENEDETTI, MS
论文数:
0
引用数:
0
h-index:
0
机构:
CHU CLERMONT FERRAND,F-63003 CLERMONT FERRAND,FRANCE
CHU CLERMONT FERRAND,F-63003 CLERMONT FERRAND,FRANCE
BENEDETTI, MS
DORDAIN, G
论文数:
0
引用数:
0
h-index:
0
机构:
CHU CLERMONT FERRAND,F-63003 CLERMONT FERRAND,FRANCE
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