(2RSTAR,3SSTAR)-1-[I-125]IODO-2,3-BIS(4-HYDROXYPHENYL)PENTANE ([I-125]IODONORHEXESTROL) AND (2RSTAR,3SSTAR)-1-[BR-77]BROMO-2,3-BIS(4-HYDROXYPHENYL)PENTANE ([BR-77]BROMONORHEXESTROL), 2 GAMMA-EMITTING ESTROGENS THAT SHOW RECEPTOR-MEDIATED UPTAKE BY TARGET TISSUES INVIVO

被引：31

作者：

LANDVATTER, SW

KATZENELLENBOGEN, JA

MCELVANY, KD

WELCH, MJ

机构：

[1] UNIV ILLINOIS,SCH CHEM SCI,URBANA,IL 61801

[2] WASHINGTON UNIV,SCH MED,EDWARD MALLINCKRODT INST RADIOL,ST LOUIS,MO 63110

[3] UNIV CALIF LOS ALAMOS NATL LAB,LOS ALAMOS,NM 87545

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1982年 / 25卷 / 11期

关键词：

D O I：

10.1021/jm00353a007

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1307 / 1312

页数：6

共 25 条

[1]

ALLEGRA JC, 1979, CANCER RES, V39, P1447

[2] NEIGHBORING CARBON AND HYDROGEN .51. DIENONES FROM ARO-3 PARTICIPATION - ISOLATION AND BEHAVIOR OF SPIRO(2,5)OCTA-1,4-DIENE-3-ONE [J].

BAIRD, R ;

WINSTEIN, S .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1963, 85 (05) :567-&

[3] FLUORINATED SULPHONIC ACIDS .1. PERFLUORO-METHANE-SULPHONIC, PERFLUORO-OCTANE-SULPHONIC, AND PERFLUORO-DECANE-SULPHONIC ACIDS AND THEIR SIMPLE DERIVATIVES [J].

BURDON, J ;

FARAZMAND, I ;

STACEY, M ;

TATLOW, JC .

JOURNAL OF THE CHEMICAL SOCIETY, 1957, (JUN) :2574-2578

[4]

CHAMNESS GC, 1978, RECEPTORS HORMONE AC, V2, P401

[5] A NEW STEREOSPECIFIC SYNTHESIS OF TRISUBSTITUTED OLEFINS . STEREOSPECIFIC SYNTHESIS OF FARNESOL [J].

COREY, EJ ;

KATZENEL.JA ;

POSNER, GH .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1967, 89 (16) :4245-&

[6]

DESPHANDE N, 1967, STEROIDS, V10, P219

[7]

FOLCA PJ, 1961, LANCET, P795

[8] ESTROGEN-RECEPTOR BASED IMAGING AGENTS .2. SYNTHESIS AND RECEPTOR-BINDING AFFINITY OF SIDE-CHAIN HALOGENATED HEXESTROL DERIVATIVES [J].

GOSWAMI, R ;

HARSY, SG ;

HEIMAN, DF ;

KATZENELLENBOGEN, JA .

JOURNAL OF MEDICINAL CHEMISTRY, 1980, 23 (09) :1002-1008

[9] THE PRODUCTION AND RECOVERY OF BR-77 AT LOS ALAMOS FOR NUCLEAR-MEDICINE STUDIES [J].

GRANT, PM ;

WHIPPLE, RE ;

BARNES, JW ;

BENTLEY, GE ;

WANEK, PM ;

OBRIEN, HA .

JOURNAL OF INORGANIC & NUCLEAR CHEMISTRY, 1981, 43 (10) :2217-2222

[10] ESTROGEN-RECEPTOR BASED IMAGING AGENTS .1. SYNTHESIS AND RECEPTOR-BINDING AFFINITY OF SOME AROMATIC AND D-RING HALOGENATED ESTROGENS [J].

HEIMAN, DF ;

SENDEROFF, SG ;

KATZENELLENBOGEN, JA ;

NEELEY, RJ .

JOURNAL OF MEDICINAL CHEMISTRY, 1980, 23 (09) :994-1002

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