A FUNDAMENTAL TEMPERATURE-DEPENDENT DIFFERENCE BETWEEN BETA-ADRENOCEPTOR AGONISTS AND ANTAGONISTS

被引:10
作者
CHESSWILLIAMS, RG
BROADLEY, KJ
DUNCAN, C
机构
关键词
D O I
10.1016/0024-3205(84)90074-2
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
引用
收藏
页码:1091 / 1099
页数:9
相关论文
共 37 条
[1]   TEMPERATURE RELATED EFFECTS ON THE BINDING CHARACTERISTICS OF BETA-ADRENERGIC-RECEPTOR AGONISTS AND ANTAGONISTS BY RABBIT LUNG [J].
ALTIERE, RJ ;
DOUGLAS, JS ;
GILLIS, CN .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1981, 316 (04) :278-287
[2]   A THEORETICAL-MODEL FOR THE USE OF FUNCTIONAL ANTAGONISM TO ESTIMATE DISSOCIATION-CONSTANTS FOR AGONISTS [J].
AMIDON, GL ;
BUCKNER, CK .
JOURNAL OF PHARMACOLOGICAL METHODS, 1982, 7 (02) :173-178
[3]   SOME QUANTITATIVE USES OF DRUG ANTAGONISTS [J].
ARUNLAKSHANA, O ;
SCHILD, HO .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1959, 14 (01) :48-58
[4]   THE EFFECT OF THE BETA-ADRENORECEPTOR ANTAGONIST RO03-7894 ON RAT ATRIAL TENSION DEVELOPMENT AND (-)-[H-3] DIHYDROALPRENOLOL BINDING TO CARDIAC AND LUNG MEMBRANES [J].
BAKER, SP ;
POSNER, P .
LIFE SCIENCES, 1983, 33 (05) :459-466
[5]   PARALLEL MODULATION OF CATECHOLAMINE ACTIVATION OF ADENYLATE-CYCLASE AND FORMATION OF THE HIGH-AFFINITY AGONIST-RECEPTOR COMPLEX IN TURKEY ERYTHROCYTE-MEMBRANES BY TEMPERATURE AND CIS-VACCENIC ACID [J].
BRIGGS, MM ;
LEFKOWITZ, RJ .
BIOCHEMISTRY, 1980, 19 (19) :4461-4466
[6]   TEMPERATURE-INDUCED CHANGES IN DISSOCIATION-CONSTANTS (KA) OF AGONISTS AT CARDIAC BETA-ADRENOCEPTORS DETERMINED BY USE OF THE IRREVERSIBLE ANTAGONIST RO-03-7894 [J].
BROADLEY, KJ ;
WILLIAMS, RG .
BRITISH JOURNAL OF PHARMACOLOGY, 1983, 79 (02) :517-524
[7]  
BROADLEY KJ, 1977, GEN PHARMACOL, V8, P305, DOI 10.1016/0306-3623(77)90004-0
[8]   DISSOCIATION-CONSTANTS (KA) AND RELATIVE EFFICACIES OF SYMPATHOMIMETIC AMINES IN ISOLATED ATRIA DURING HYPOTHERMIA-INDUCED SUPER-SENSITIVITY [J].
BROADLEY, KJ ;
MCNEILL, JH .
CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY, 1983, 61 (06) :572-580
[9]   FUNCTIONAL ANTAGONISM AS A MEANS OF DETERMINING DISSOCIATION-CONSTANTS AND RELATIVE EFFICACIES OF SYMPATHOMIMETIC AMINES IN GUINEA-PIG ISOLATED ATRIA [J].
BROADLEY, KJ ;
NICHOLSON, CD .
BRITISH JOURNAL OF PHARMACOLOGY, 1979, 66 (03) :397-404
[10]  
BROADLEY KJ, 1980, METHOD FIND EXP CLIN, V2, P181