A COMPARISON OF 2 CYTO-TOXICITY ASSAYS FOR THE DETECTION OF METABOLISM-MEDIATED TOXICITY INVITRO - A STUDY WITH CYCLOPHOSPHAMIDE

被引:18
作者
HORNER, SA [1 ]
FRY, JR [1 ]
CLOTHIER, RH [1 ]
BALLS, M [1 ]
机构
[1] UNIV NOTTINGHAM HOSP,QUEENS MED CTR,SCH MED,DEPT PHYSIOL & PHARMACOL,NOTTINGHAM NG7 2UH,ENGLAND
关键词
D O I
10.3109/00498258509047427
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:681 / 686
页数:6
相关论文
共 21 条
[1]   METABOLIC-ACTIVATION AND CYTO-TOXICITY OF CYCLOPHOSPHAMIDE IN PRIMARY CULTURES OF POSTNATAL RAT HEPATOCYTES [J].
ACOSTA, D ;
MITCHELL, DB .
BIOCHEMICAL PHARMACOLOGY, 1981, 30 (23) :3225-3230
[2]  
CONNEY AH, 1982, CANCER RES, V42, P4875
[3]   TOXICITY TESTING INVITRO .2. USE OF A MICROSOME-CULTURED HUMAN FIBROBLAST SYSTEM TO STUDY CYTOTOXICITY OF CYCLOPHOSPHAMIDE [J].
COOPER, JT ;
GOLDSTEIN, S .
CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY, 1976, 54 (04) :546-550
[4]  
COX PJ, 1975, CANCER RES, V35, P3755
[5]  
HALES BF, 1982, CANCER RES, V42, P3016
[6]   CHARACTERISTICS OF THE ACTIVATION OF CYCLOPHOSPHAMIDE TO A MUTAGEN BY RAT-LIVER [J].
HALES, BF ;
JAIN, R .
BIOCHEMICAL PHARMACOLOGY, 1980, 29 (02) :256-259
[7]  
HORNER SA, 1984, ATLA, V11, P147
[8]   CELL-MEDIATED MUTAGENESIS OF MAMMALIAN-CELLS WITH CHEMICAL CARCINOGENS [J].
HUBERMAN, E ;
SACHS, L .
INTERNATIONAL JOURNAL OF CANCER, 1974, 13 (03) :326-333
[9]   SEX DIFFERENCE IN THE O-DEALKYLATION ACTIVITY OF 7-HYDROXYCOUMARIN O-ALKYL DERIVATIVES IN LIVER-MICROSOMES OF RATS [J].
KAMATAKI, T ;
ANDO, M ;
YAMAZOE, Y ;
ISHII, K ;
KATO, R .
BIOCHEMICAL PHARMACOLOGY, 1980, 29 (07) :1015-1022
[10]   LIVER HOMOGENATE-MEDIATED MUTAGENESIS IN CHINESE-HAMSTER V79 CELLS BY POLYCYCLIC AROMATIC-HYDROCARBONS AND AFLATOXINS [J].
KRAHN, DF ;
HEIDELBERGER, C .
MUTATION RESEARCH, 1977, 46 (01) :27-44