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ORALLY ACTIVE AND POTENT INHIBITORS OF GAMMA-AMINOBUTYRIC ACID UPTAKE
被引:135
作者
:
ALI, FE
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DIV RES & DEV,DEPT MED CHEM,PHILADELPHIA,PA 19101
ALI, FE
BONDINELL, WE
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DIV RES & DEV,DEPT MED CHEM,PHILADELPHIA,PA 19101
BONDINELL, WE
DANDRIDGE, PA
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DIV RES & DEV,DEPT MED CHEM,PHILADELPHIA,PA 19101
DANDRIDGE, PA
FRAZEE, JS
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DIV RES & DEV,DEPT MED CHEM,PHILADELPHIA,PA 19101
FRAZEE, JS
GARVEY, E
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DIV RES & DEV,DEPT MED CHEM,PHILADELPHIA,PA 19101
GARVEY, E
GIRARD, GR
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DIV RES & DEV,DEPT MED CHEM,PHILADELPHIA,PA 19101
GIRARD, GR
KAISER, C
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DIV RES & DEV,DEPT MED CHEM,PHILADELPHIA,PA 19101
KAISER, C
KU, TW
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DIV RES & DEV,DEPT MED CHEM,PHILADELPHIA,PA 19101
KU, TW
LAFFERTY, JJ
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DIV RES & DEV,DEPT MED CHEM,PHILADELPHIA,PA 19101
LAFFERTY, JJ
MOONSAMMY, GI
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DIV RES & DEV,DEPT MED CHEM,PHILADELPHIA,PA 19101
MOONSAMMY, GI
OH, HJ
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DIV RES & DEV,DEPT MED CHEM,PHILADELPHIA,PA 19101
OH, HJ
RUSH, JA
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DIV RES & DEV,DEPT MED CHEM,PHILADELPHIA,PA 19101
RUSH, JA
SETLER, PE
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DIV RES & DEV,DEPT MED CHEM,PHILADELPHIA,PA 19101
SETLER, PE
STRINGER, OD
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DIV RES & DEV,DEPT MED CHEM,PHILADELPHIA,PA 19101
STRINGER, OD
VENSLAVSKY, JW
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DIV RES & DEV,DEPT MED CHEM,PHILADELPHIA,PA 19101
VENSLAVSKY, JW
VOLPE, BW
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DIV RES & DEV,DEPT MED CHEM,PHILADELPHIA,PA 19101
VOLPE, BW
YUNGER, LM
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DIV RES & DEV,DEPT MED CHEM,PHILADELPHIA,PA 19101
YUNGER, LM
ZIRKLE, CL
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F LABS,DIV RES & DEV,DEPT MED CHEM,PHILADELPHIA,PA 19101
ZIRKLE, CL
机构
:
[1]
SK&F LABS,DIV RES & DEV,DEPT MED CHEM,PHILADELPHIA,PA 19101
[2]
SK&F LABS,DIV RES & DEV,DEPT PHARMACOL,PHILADELPHIA,PA 19101
来源
:
JOURNAL OF MEDICINAL CHEMISTRY
|
1985年
/ 28卷
/ 05期
关键词
:
D O I
:
10.1021/jm50001a020
中图分类号
:
R914 [药物化学];
学科分类号
:
100701 ;
摘要
:
引用
收藏
页码:653 / 660
页数:8
相关论文
共 64 条
[1]
ALBERT A, 1971, DETERMINATION IONIZA
[2]
SYNTHETIC ANALOGS FOR THE STUDY OF GABA AS A NEUROTRANSMITTER
ALLAN, RD
论文数:
0
引用数:
0
h-index:
0
ALLAN, RD
JOHNSTON, GAR
论文数:
0
引用数:
0
h-index:
0
JOHNSTON, GAR
[J].
MEDICINAL RESEARCH REVIEWS,
1983,
3
(02)
: 91
-
118
[3]
MUSCIMOL AND RELATED GABA RECEPTOR AGONISTS - POTENCY OF GABAERGIC DRUGS INVIVO DETERMINED AFTER INTRANIGRAL INJECTION
ARNT, J
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT PHARMACOL, DK-2100 COPENHAGEN, DENMARK
ARNT, J
SCHEELKRUGER, J
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT PHARMACOL, DK-2100 COPENHAGEN, DENMARK
SCHEELKRUGER, J
MAGELUND, G
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT PHARMACOL, DK-2100 COPENHAGEN, DENMARK
MAGELUND, G
KROGSGAARDLARSEN, P
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT PHARMACOL, DK-2100 COPENHAGEN, DENMARK
KROGSGAARDLARSEN, P
[J].
JOURNAL OF PHARMACY AND PHARMACOLOGY,
1979,
31
(05)
: 306
-
313
[4]
GABA IN THE OLFACTORY-BULB AND OLFACTORY NUCLEUS OF THE RAT - DISTRIBUTION OF GAMMA-AMINOBUTYRIC ACID, GLUTAMIC-ACID DECARBOXYLASE, GABA TRANSAMINASE AND SUCCINATE SEMI-ALDEHYDE DEHYDROGENASE
AUSTIN, L
论文数:
0
引用数:
0
h-index:
0
机构:
CNRS,CTR NEUROCHIM,INST CHIM BIOL,F-67085 STRASBOURG,FRANCE
CNRS,CTR NEUROCHIM,INST CHIM BIOL,F-67085 STRASBOURG,FRANCE
AUSTIN, L
RECASENS, M
论文数:
0
引用数:
0
h-index:
0
机构:
CNRS,CTR NEUROCHIM,INST CHIM BIOL,F-67085 STRASBOURG,FRANCE
CNRS,CTR NEUROCHIM,INST CHIM BIOL,F-67085 STRASBOURG,FRANCE
RECASENS, M
MANDEL, P
论文数:
0
引用数:
0
h-index:
0
机构:
CNRS,CTR NEUROCHIM,INST CHIM BIOL,F-67085 STRASBOURG,FRANCE
CNRS,CTR NEUROCHIM,INST CHIM BIOL,F-67085 STRASBOURG,FRANCE
MANDEL, P
[J].
JOURNAL OF NEUROCHEMISTRY,
1979,
32
(05)
: 1473
-
1477
[5]
CHARACTERISTICS OF GABAB RECEPTOR-BINDING SITES ON RAT WHOLE BRAIN SYNAPTIC-MEMBRANES
BOWERY, NG
论文数:
0
引用数:
0
h-index:
0
BOWERY, NG
HILL, DR
论文数:
0
引用数:
0
h-index:
0
HILL, DR
HUDSON, AL
论文数:
0
引用数:
0
h-index:
0
HUDSON, AL
[J].
BRITISH JOURNAL OF PHARMACOLOGY,
1983,
78
(01)
: 191
-
206
[6]
SELECTIVE-INHIBITION OF NEURONAL GABA UPTAKE BY CIS-1,3-AMINOCYCLOHEXANE CARBOXYLIC-ACID
BOWERY, NG
论文数:
0
引用数:
0
h-index:
0
机构:
ST THOMAS HOSP & MED SCH, SCH MED, DEPT PHARMACOL, LONDON SE1 7EH, ENGLAND
BOWERY, NG
JONES, GP
论文数:
0
引用数:
0
h-index:
0
机构:
ST THOMAS HOSP & MED SCH, SCH MED, DEPT PHARMACOL, LONDON SE1 7EH, ENGLAND
JONES, GP
NEAL, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
ST THOMAS HOSP & MED SCH, SCH MED, DEPT PHARMACOL, LONDON SE1 7EH, ENGLAND
NEAL, MJ
[J].
NATURE,
1976,
264
(5583)
: 281
-
284
[7]
ESTERS OF NIPECOTIC AND ISONIPECOTIC ACIDS AS POTENTIAL ANTICONVULSANTS
CRIDER, AM
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV SASKATCHEWAN,DEPT BIOCHEM,SASKATOON S7N 0W0,SASKATCHEWAN,CANADA
UNIV SASKATCHEWAN,DEPT BIOCHEM,SASKATOON S7N 0W0,SASKATCHEWAN,CANADA
CRIDER, AM
TITA, TT
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV SASKATCHEWAN,DEPT BIOCHEM,SASKATOON S7N 0W0,SASKATCHEWAN,CANADA
UNIV SASKATCHEWAN,DEPT BIOCHEM,SASKATOON S7N 0W0,SASKATCHEWAN,CANADA
TITA, TT
WOOD, JD
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV SASKATCHEWAN,DEPT BIOCHEM,SASKATOON S7N 0W0,SASKATCHEWAN,CANADA
UNIV SASKATCHEWAN,DEPT BIOCHEM,SASKATOON S7N 0W0,SASKATCHEWAN,CANADA
WOOD, JD
HINKO, CN
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV SASKATCHEWAN,DEPT BIOCHEM,SASKATOON S7N 0W0,SASKATCHEWAN,CANADA
UNIV SASKATCHEWAN,DEPT BIOCHEM,SASKATOON S7N 0W0,SASKATCHEWAN,CANADA
HINKO, CN
[J].
JOURNAL OF PHARMACEUTICAL SCIENCES,
1982,
71
(11)
: 1214
-
1219
[8]
ANTI-CONVULSANT ACTIVITY OF GABA UPTAKE INHIBITORS AND THEIR PRODRUGS FOLLOWING CENTRAL OR SYSTEMIC ADMINISTRATION
CROUCHER, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
KINGS COLL HOSP MED SCH,RAYNE INST,DEPT NEUROL,LONDON SE5 9NU,ENGLAND
CROUCHER, MJ
MELDRUM, BS
论文数:
0
引用数:
0
h-index:
0
机构:
KINGS COLL HOSP MED SCH,RAYNE INST,DEPT NEUROL,LONDON SE5 9NU,ENGLAND
MELDRUM, BS
KROGSGAARDLARSEN, P
论文数:
0
引用数:
0
h-index:
0
机构:
KINGS COLL HOSP MED SCH,RAYNE INST,DEPT NEUROL,LONDON SE5 9NU,ENGLAND
KROGSGAARDLARSEN, P
[J].
EUROPEAN JOURNAL OF PHARMACOLOGY,
1983,
89
(3-4)
: 217
-
228
[9]
CURTIS DR, 1979, GABA NEUROTRANSMITTE, P17
[10]
NEW PSYCHOTROPIC AGENTS .8. ANALOGS OF AMITRIPTYLINE CONTAINING NORMEPERIDINE GROUP
DAVIS, MA
论文数:
0
引用数:
0
h-index:
0
DAVIS, MA
HERR, F
论文数:
0
引用数:
0
h-index:
0
HERR, F
THOMAS, RA
论文数:
0
引用数:
0
h-index:
0
THOMAS, RA
CHAREST, MP
论文数:
0
引用数:
0
h-index:
0
CHAREST, MP
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1967,
10
(04)
: 627
-
&
←
1
2
3
4
5
6
7
→
共 64 条
[1]
ALBERT A, 1971, DETERMINATION IONIZA
[2]
SYNTHETIC ANALOGS FOR THE STUDY OF GABA AS A NEUROTRANSMITTER
ALLAN, RD
论文数:
0
引用数:
0
h-index:
0
ALLAN, RD
JOHNSTON, GAR
论文数:
0
引用数:
0
h-index:
0
JOHNSTON, GAR
[J].
MEDICINAL RESEARCH REVIEWS,
1983,
3
(02)
: 91
-
118
[3]
MUSCIMOL AND RELATED GABA RECEPTOR AGONISTS - POTENCY OF GABAERGIC DRUGS INVIVO DETERMINED AFTER INTRANIGRAL INJECTION
ARNT, J
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT PHARMACOL, DK-2100 COPENHAGEN, DENMARK
ARNT, J
SCHEELKRUGER, J
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT PHARMACOL, DK-2100 COPENHAGEN, DENMARK
SCHEELKRUGER, J
MAGELUND, G
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT PHARMACOL, DK-2100 COPENHAGEN, DENMARK
MAGELUND, G
KROGSGAARDLARSEN, P
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL DANISH SCH PHARM, DEPT PHARMACOL, DK-2100 COPENHAGEN, DENMARK
KROGSGAARDLARSEN, P
[J].
JOURNAL OF PHARMACY AND PHARMACOLOGY,
1979,
31
(05)
: 306
-
313
[4]
GABA IN THE OLFACTORY-BULB AND OLFACTORY NUCLEUS OF THE RAT - DISTRIBUTION OF GAMMA-AMINOBUTYRIC ACID, GLUTAMIC-ACID DECARBOXYLASE, GABA TRANSAMINASE AND SUCCINATE SEMI-ALDEHYDE DEHYDROGENASE
AUSTIN, L
论文数:
0
引用数:
0
h-index:
0
机构:
CNRS,CTR NEUROCHIM,INST CHIM BIOL,F-67085 STRASBOURG,FRANCE
CNRS,CTR NEUROCHIM,INST CHIM BIOL,F-67085 STRASBOURG,FRANCE
AUSTIN, L
RECASENS, M
论文数:
0
引用数:
0
h-index:
0
机构:
CNRS,CTR NEUROCHIM,INST CHIM BIOL,F-67085 STRASBOURG,FRANCE
CNRS,CTR NEUROCHIM,INST CHIM BIOL,F-67085 STRASBOURG,FRANCE
RECASENS, M
MANDEL, P
论文数:
0
引用数:
0
h-index:
0
机构:
CNRS,CTR NEUROCHIM,INST CHIM BIOL,F-67085 STRASBOURG,FRANCE
CNRS,CTR NEUROCHIM,INST CHIM BIOL,F-67085 STRASBOURG,FRANCE
MANDEL, P
[J].
JOURNAL OF NEUROCHEMISTRY,
1979,
32
(05)
: 1473
-
1477
[5]
CHARACTERISTICS OF GABAB RECEPTOR-BINDING SITES ON RAT WHOLE BRAIN SYNAPTIC-MEMBRANES
BOWERY, NG
论文数:
0
引用数:
0
h-index:
0
BOWERY, NG
HILL, DR
论文数:
0
引用数:
0
h-index:
0
HILL, DR
HUDSON, AL
论文数:
0
引用数:
0
h-index:
0
HUDSON, AL
[J].
BRITISH JOURNAL OF PHARMACOLOGY,
1983,
78
(01)
: 191
-
206
[6]
SELECTIVE-INHIBITION OF NEURONAL GABA UPTAKE BY CIS-1,3-AMINOCYCLOHEXANE CARBOXYLIC-ACID
BOWERY, NG
论文数:
0
引用数:
0
h-index:
0
机构:
ST THOMAS HOSP & MED SCH, SCH MED, DEPT PHARMACOL, LONDON SE1 7EH, ENGLAND
BOWERY, NG
JONES, GP
论文数:
0
引用数:
0
h-index:
0
机构:
ST THOMAS HOSP & MED SCH, SCH MED, DEPT PHARMACOL, LONDON SE1 7EH, ENGLAND
JONES, GP
NEAL, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
ST THOMAS HOSP & MED SCH, SCH MED, DEPT PHARMACOL, LONDON SE1 7EH, ENGLAND
NEAL, MJ
[J].
NATURE,
1976,
264
(5583)
: 281
-
284
[7]
ESTERS OF NIPECOTIC AND ISONIPECOTIC ACIDS AS POTENTIAL ANTICONVULSANTS
CRIDER, AM
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV SASKATCHEWAN,DEPT BIOCHEM,SASKATOON S7N 0W0,SASKATCHEWAN,CANADA
UNIV SASKATCHEWAN,DEPT BIOCHEM,SASKATOON S7N 0W0,SASKATCHEWAN,CANADA
CRIDER, AM
TITA, TT
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV SASKATCHEWAN,DEPT BIOCHEM,SASKATOON S7N 0W0,SASKATCHEWAN,CANADA
UNIV SASKATCHEWAN,DEPT BIOCHEM,SASKATOON S7N 0W0,SASKATCHEWAN,CANADA
TITA, TT
WOOD, JD
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV SASKATCHEWAN,DEPT BIOCHEM,SASKATOON S7N 0W0,SASKATCHEWAN,CANADA
UNIV SASKATCHEWAN,DEPT BIOCHEM,SASKATOON S7N 0W0,SASKATCHEWAN,CANADA
WOOD, JD
HINKO, CN
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV SASKATCHEWAN,DEPT BIOCHEM,SASKATOON S7N 0W0,SASKATCHEWAN,CANADA
UNIV SASKATCHEWAN,DEPT BIOCHEM,SASKATOON S7N 0W0,SASKATCHEWAN,CANADA
HINKO, CN
[J].
JOURNAL OF PHARMACEUTICAL SCIENCES,
1982,
71
(11)
: 1214
-
1219
[8]
ANTI-CONVULSANT ACTIVITY OF GABA UPTAKE INHIBITORS AND THEIR PRODRUGS FOLLOWING CENTRAL OR SYSTEMIC ADMINISTRATION
CROUCHER, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
KINGS COLL HOSP MED SCH,RAYNE INST,DEPT NEUROL,LONDON SE5 9NU,ENGLAND
CROUCHER, MJ
MELDRUM, BS
论文数:
0
引用数:
0
h-index:
0
机构:
KINGS COLL HOSP MED SCH,RAYNE INST,DEPT NEUROL,LONDON SE5 9NU,ENGLAND
MELDRUM, BS
KROGSGAARDLARSEN, P
论文数:
0
引用数:
0
h-index:
0
机构:
KINGS COLL HOSP MED SCH,RAYNE INST,DEPT NEUROL,LONDON SE5 9NU,ENGLAND
KROGSGAARDLARSEN, P
[J].
EUROPEAN JOURNAL OF PHARMACOLOGY,
1983,
89
(3-4)
: 217
-
228
[9]
CURTIS DR, 1979, GABA NEUROTRANSMITTE, P17
[10]
NEW PSYCHOTROPIC AGENTS .8. ANALOGS OF AMITRIPTYLINE CONTAINING NORMEPERIDINE GROUP
DAVIS, MA
论文数:
0
引用数:
0
h-index:
0
DAVIS, MA
HERR, F
论文数:
0
引用数:
0
h-index:
0
HERR, F
THOMAS, RA
论文数:
0
引用数:
0
h-index:
0
THOMAS, RA
CHAREST, MP
论文数:
0
引用数:
0
h-index:
0
CHAREST, MP
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1967,
10
(04)
: 627
-
&
←
1
2
3
4
5
6
7
→