ENALAPRIL MALEATE (MK-421), A POTENT, NONSULFHYDRYL ANGIOTENSIN-CONVERTING ENZYME-INHIBITOR - ABSORPTION, DISPOSITION, AND METABOLISM IN MAN

被引:83
作者
ULM, EH
机构
关键词
D O I
10.3109/03602538308991383
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:99 / 110
页数:12
相关论文
共 18 条
  • [1] ANDERSON T, 1981, NEW ENGL J MED, V304, P1550
  • [2] 3 NEW LONG-ACTING CONVERTING-ENZYME INHIBITORS - RELATIONSHIP BETWEEN PLASMA CONVERTING-ENZYME ACTIVITY AND RESPONSE TO ANGIOTENSIN-I
    BIOLLAZ, J
    BURNIER, M
    TURINI, GA
    BRUNNER, DB
    PORCHET, M
    GOMEZ, HJ
    JONES, KH
    FERBER, F
    ABRAMS, WB
    GAVRAS, H
    BRUNNER, HR
    [J]. CLINICAL PHARMACOLOGY & THERAPEUTICS, 1981, 29 (05) : 665 - 670
  • [3] BIOLLAZ J, BR J CLIN PHARM
  • [4] EFFECT OF A NEW ANGIOTENSIN CONVERTING ENZYME-INHIBITOR MK 421 AND ITS LYSINE ANALOG ON THE COMPONENTS OF THE RENIN SYSTEM IN HEALTHY-SUBJECTS
    BRUNNER, DB
    DESPONDS, G
    BIOLLAZ, J
    KELLER, I
    FERBER, F
    GAVRAS, H
    BRUNNER, HR
    SCHELLING, JL
    [J]. BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1981, 11 (05) : 461 - 467
  • [5] Cushman D W, 1980, Prog Med Chem, V17, P41, DOI 10.1016/S0079-6468(08)70157-7
  • [6] DAVIS JO, 1976, PHYSL REV, V15, P1
  • [7] GROSS DM, 1981, J PHARMACOL EXP THER, V216, P552
  • [8] HICHENS M, 1981, Ligand Quarterly, V4, P43
  • [9] LAFFAN RJ, 1978, J PHARMACOL EXP THER, V204, P281
  • [10] DESIGN OF SPECIFIC INHIBITORS OF ANGIOTENSIN-CONVERTING ENZYME - NEW CLASS OF ORALLY ACTIVE ANTIHYPERTENSIVE AGENTS
    ONDETTI, MA
    CUSHMAN, DW
    [J]. SCIENCE, 1977, 196 (4288) : 441 - 444