DISCOVERY OF ALTERED PHARMACOKINETICS OF CGP 15 210 G IN POOR HYDROXYLATORS OF DEBRISOQUINE DURING EARLY DRUG DEVELOPMENT

被引:7
作者
GLEITER, CH
AICHELE, G
NILSSON, E
HENGEN, N
ANTONIN, KH
BIECK, PR
机构
关键词
D O I
10.1111/j.1365-2125.1985.tb02802.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
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页码:81 / 84
页数:4
相关论文
共 10 条
[1]  
ANTONIN K H, 1984, Naunyn-Schmiedeberg's Archives of Pharmacology, V325, pR90
[2]  
DICK B, 1982, SCHWEIZ MED WSCHR, V112, P1061
[3]   A FAMILY AND POPULATION STUDY OF THE GENETIC-POLYMORPHISM OF DEBRISOQUINE OXIDATION IN A WHITE BRITISH-POPULATION [J].
EVANS, DAP ;
MAHGOUB, A ;
SLOAN, TP ;
IDLE, JR ;
SMITH, RL .
JOURNAL OF MEDICAL GENETICS, 1980, 17 (02) :102-105
[4]   POLYMORPHISMS OF OXIDATION AT CARBON CENTERS OF DRUGS AND THEIR CLINICAL SIGNIFICANCE [J].
IDLE, JR ;
SMITH, RL .
DRUG METABOLISM REVIEWS, 1979, 9 (02) :301-317
[5]  
IDLE JR, 1983, LANCET, V1, P1388
[6]   DETERMINATION OF DEBRISOQUINE AND ITS 4-HYDROXY METABOLITE IN BIOLOGICAL-FLUIDS BY GAS-CHROMATOGRAPHY WITH FLAME-IONIZATION AND NITROGEN-SELECTIVE DETECTION [J].
LENNARD, MS ;
SILAS, JH ;
SMITH, AJ ;
TUCKER, GT .
JOURNAL OF CHROMATOGRAPHY, 1977, 133 (01) :161-166
[7]  
LENNARD MS, 1984, BRIT J CLIN PHARMACO, V17, P489
[8]   POLYMORPHIC HYDROXYLATION OF DEBRISOQUINE IN MAN [J].
MAHGOUB, A ;
IDLE, JR ;
DRING, LG ;
LANCASTER, R ;
SMITH, RL .
LANCET, 1977, 2 (8038) :584-586
[9]  
RITSCHEL WA, 1980, HDB BASIC PHARMACOKI, P208
[10]  
SCHNEIDER W, 1982, DETERMINATION UNCHAN