SYNTHESIS OF NEW TAXOIDS

被引：15

作者：

BLECHERT, S

JANSEN, R

VELDER, J

机构：

[1] Technische Universität Berlin, D-10623 Berlin

来源：

TETRAHEDRON | 1994年 / 50卷 / 32期

关键词：

D O I：

10.1016/S0040-4020(01)85533-2

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

[2+2] Photocycloadditions between enone 2 and 2,3-dihydropyran derivatives lead to a number of interesting intermediates 3a-e for taxoid synthesis. Following this strategy the stereoselective synthesis of a biologically active taxoid mimicking the polarity of the CD ring portion in taxol is reported.

引用

收藏

页码：9649 / 9656

页数：8

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