PHYSIOLOGICALLY BASED PHARMACOKINETIC MODEL FOR BETA-LACTAM ANTIBIOTICS-I - TISSUE DISTRIBUTION AND ELIMINATION IN RATS

被引:153
作者
TSUJI, A
YOSHIKAWA, T
NISHIDE, K
MINAMI, H
KIMURA, M
NAKASHIMA, E
TERASAKI, T
MIYAMOTO, E
NIGHTINGALE, CH
YAMANA, T
机构
[1] HARTFORD HOSP, HARTFORD, CT 06115 USA
[2] UNIV CONNECTICUT, SCH PHARM, STORRS, CT 06268 USA
关键词
D O I
10.1002/jps.2600721103
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
收藏
页码:1239 / 1252
页数:14
相关论文
共 61 条
[11]   TRANSPORT AND BINDING OF METHOTREXATE IN-VIVO [J].
DEDRICK, RL ;
ZAHARKO, DS ;
LUTZ, RJ .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1973, 62 (06) :882-890
[12]  
DINGELDEIN E, 1979, ARZNEIMITTEL-FORSCH, V29-2, P400
[13]  
DITTERT LW, 1970, ANTIMICROB AGENTS CH, P42
[14]  
ENGLISH AR, 1960, P SOC EXP BIOL MED, V104, P405, DOI 10.3181/00379727-104-25853
[15]  
GIBALDI M, 1969, ANTIMICROB AGENTS CH, P378
[16]   BINDING RATE OF ANTIBACTERIALS TO SERUM-PROTEINS [J].
GREENE, DS ;
QUINTILIANI, R ;
NIGHTINGALE, CH .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1977, 66 (11) :1663-1664
[17]   PHYSIOLOGICAL PERFUSION MODEL FOR CEPHALOSPORIN ANTIBIOTICS .1. MODEL SELECTION BASED ON BLOOD DRUG CONCENTRATIONS [J].
GREENE, DS ;
QUINTILIANI, R ;
NIGHTINGALE, CH .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1978, 67 (02) :191-196
[18]   DETERMINATION OF PROBENECID IN SERUM BY HIGH-PERFORMANCE LIQUID-CHROMATOGRAPHY [J].
HARLE, RK ;
COWEN, T .
ANALYST, 1978, 103 (1226) :492-496
[19]   PHYSIOLOGICALLY BASED PHARMACOKINETIC MODEL FOR DIGOXIN DISPOSITION IN DOGS AND ITS PRELIMINARY APPLICATION TO HUMANS [J].
HARRISON, LI ;
GIBALDI, M .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1977, 66 (12) :1679-1683
[20]  
HIGAKI K, 1969, Journal of the Physiological Society of Japan, V31, P164