MIXED COMPETITIVE AND ALLOSTERIC ANTAGONISM BY GALLAMINE OF MUSCARINIC RECEPTOR-MEDIATED 2ND MESSENGER RESPONSES IN N1E-115 NEURO-BLASTOMA CELLS

被引:18
作者
LEE, NH [1 ]
ELFAKAHANY, EE [1 ]
机构
[1] UNIV MARYLAND,SCH PHARM,DEPT PHARMACOL & TOXICOL,20 N PINE ST,BALTIMORE,MD 21201
关键词
D O I
10.1111/j.1471-4159.1989.tb07428.x
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:1300 / 1308
页数:9
相关论文
共 52 条
[11]   INTERACTIONS OF QUINIDINE AND LIDOCAINE WITH RAT-BRAIN AND HEART MUSCARINIC RECEPTORS [J].
COHEN-ARMON, M ;
HENIS, YI ;
KLOOG, Y ;
SOKOLOVSKY, M .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1985, 127 (01) :326-332
[12]  
DOODS HN, 1987, J PHARMACOL EXP THER, V242, P257
[13]  
DUNLAP J, 1983, MOL PHARMACOL, V24, P15
[14]   COMPETITIVE AND NONCOMPETITIVE ANTAGONISM EXHIBITED BY SELECTIVE ANTAGONISTS AT ATRIAL AND ILEAL MUSCARINIC RECEPTOR SUBTYPES [J].
EGLEN, RM ;
WHITING, RL .
BRITISH JOURNAL OF PHARMACOLOGY, 1987, 90 (04) :701-707
[15]  
EHLERT FJ, 1988, MOL PHARMACOL, V33, P187
[16]  
ELFAKAHANY EE, 1984, J PHARMACOL EXP THER, V229, P447
[17]   CHARACTERIZATION OF THE INTERACTIONS OF GALLAMINE WITH MUSCARINIC RECEPTORS FROM BRAIN [J].
ELLIS, J ;
LENOX, RH .
BIOCHEMICAL PHARMACOLOGY, 1985, 34 (12) :2214-2217
[18]  
FISHER SK, 1987, MOL PHARMACOL, V32, P81
[19]  
GARDNER AL, 1988, TRENDS PHARM SCI S, V3, P40
[20]  
GIRALDO E, 1988, J PHARMACOL EXP THER, V244, P1016