PROBES FOR NARCOTIC RECEPTOR MEDIATED PHENOMENA .8. TRITIATION OF IRREVERSIBLE MU-SPECIFIC OR DELTA-SPECIFIC OPIOID RECEPTOR AFFINITY LIGANDS TO HIGH SPECIFIC ACTIVITY

被引：11

作者：

BURKE, TR ^{[1
]}

RICE, KC ^{[1
]}

JACOBSON, AE ^{[1
]}

SIMONDS, WF ^{[1
]}

KLEE, WA ^{[1
]}

机构：

[1] NIMH,GEN & COMPARAT BIOCHEM LAB,BETHESDA,MD 20205

来源：

JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS | 1984年 / 21卷 / 08期

关键词：

D O I：

10.1002/jlcr.2580210802

中图分类号：

Q5 [生物化学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：693 / 702

页数：10

共 13 条

[1]

BURKE TR, 1984, J MED CHEM

[2] IDENTIFICATION OF 2 RELATED PENTAPEPTIDES FROM BRAIN WITH POTENT OPIATE AGONIST ACTIVITY [J].

HUGHES, J ;

SMITH, TW ;

KOSTERLITZ, HW ;

FOTHERGILL, LA ;

MORGAN, BA ;

MORRIS, HR .

NATURE, 1975, 258 (5536) :577-579

[3] REACTIONS OF HETEROCYCLES WITH THIOPHOSGENE .4. BETA,4-DICHLORO-2-ISOTHIOCYANATOCINNAMALDEHYDE, A PRODUCT FROM 4,7-DICHLOROQUINOLINE [J].

HULL, R ;

VANDENBROEK, PJ ;

SWAIN, ML .

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 1975, (10) :922-925

[4] PROBES FOR NARCOTIC RECEPTOR MEDIATED PHENOMENA .5. NARCOTIC-ANTAGONIST IRREVERSIBLE LIGANDS BASED ON ENDOETHENOTETRAHYDROORIPAVINE [J].

JACOBSON, AE ;

BAJWA, BS ;

STREATY, RA ;

KLEE, WA ;

RICE, KC .

LIFE SCIENCES, 1983, 33 :159-162

[5] IDENTIFICATION OF A MR 58000 GLYCOPROTEIN SUBUNIT OF THE OPIATE RECEPTOR [J].

KLEE, WA ;

SIMONDS, WF ;

SWEAT, FW ;

BURKE, TR ;

JACOBSON, AE ;

RICE, KC .

FEBS LETTERS, 1982, 150 (01) :125-128

[6]

MARTIN WR, 1967, PHARMACOL REV, V19, P463

[7] OPIATE RECEPTOR - DEMONSTRATION IN NERVOUS-TISSUE [J].

PERT, CB ;

SNYDER, SH .

SCIENCE, 1973, 179 (4077) :1011-1014

[8] DEMONSTRATION AND DISTRIBUTION OF AN OPIATE BINDING-SITE IN RAT-BRAIN WITH HIGH-AFFINITY FOR ETHYLKETOCYCLAZOCINE AND SKF 10,047 [J].

PFEIFFER, A ;

HERZ, A .

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1981, 101 (01) :38-44

[9] IRREVERSIBLE LIGANDS WITH HIGH SELECTIVITY TOWARD DELTA-OPIATE OR MU-OPIATE RECEPTORS [J].

RICE, KC ;

JACOBSON, AE ;

BURKE, TR ;

BAJWA, BS .

SCIENCE, 1983, 220 (4594) :314-316

[10] STEREOSPECIFIC BINDING OF POTENT NARCOTIC ANALGESIC [H-3)ETORPHINE TO RAT-BRAIN HOMOGENATE [J].

SIMON, EJ ;

HILLER, JM ;

EDELMAN, I .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1973, 70 (07) :1947-1949

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