ON THE DEFINITION OF EFFICACY

被引:15
作者
KENAKIN, T
机构
关键词
D O I
10.1016/0165-6147(94)90086-8
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:408 / 409
页数:2
相关论文
共 14 条
[1]  
ARIENS EJ, 1954, ARCH INT PHARMACOD T, V99, P32
[2]  
BOND RA, 1994, CAN J PHYSL PHARM S1, V22
[3]  
CHIDIAC P, 1994, MOL PHARMACOL, V45, P490
[4]  
Colquhoun D., 1987, PERSPECTIVES RECEPTO, V6, P103
[5]   ANTAGONISTS WITH NEGATIVE INTRINSIC ACTIVITY AT DELTA-OPIOID RECEPTORS COUPLED TO GTP-BINDING PROTEINS [J].
COSTA, T ;
HERZ, A .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1989, 86 (19) :7321-7325
[6]  
COSTA T, 1992, MOL PHARMACOL, V41, P549
[7]  
DELEAN A, 1982, MOL PHARMACOL, V22, P290
[8]  
KENAKIN TP, 1992, PHARMACOL REV, V44, P351
[9]   CONSTITUTIVE ACTIVITY OF RECEPTORS COUPLED TO GUANINE-NUCLEOTIDE REGULATORY PROTEINS [J].
LEFKOWITZ, RJ ;
COTECCHIA, S ;
SAMAMA, P ;
COSTA, T .
TRENDS IN PHARMACOLOGICAL SCIENCES, 1993, 14 (08) :303-307
[10]  
SAMAMA P, 1993, J BIOL CHEM, V268, P4625