A NEW METHOD FOR THE CONSTRUCTION OF INDOLE NUCLEUS

被引：15

作者：

IWAO, M

机构：

[1] Department of Chemistry, Faculty of Liberal Arts, Nagasaki University, Nagasaki, 852

来源：

HETEROCYCLES | 1994年 / 38卷 / 01期

关键词：

D O I：

10.3987/COM-93-6563

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Directed lithiation of N-tert-butoxycarbonylanilines and subsequent reaction with 1-tert-butyldimethylsilyl-1-phenylsulfinylethene gave the conjugate addition products which, without isolation, were cyclized to 1-tert-butoxycarbonyl-2-phenylthioindolines under thermal sila-Pummerer reaction conditions.

引用

页码：45 / 50

页数：6

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