DIRECT INHIBITION OF TESTICULAR STEROIDOGENESIS AND GONADOTROPIN RECEPTOR LEVELS BY [(IMBZL)-D-HIS6,PRO9-NET]GNRH AND [D-TRP6,PRO9-NET]GNRH, POTENT AGONISTS OF GNRH

被引:25
作者
CAO, YQ
SUNDARAM, K
BARDIN, CW
RIVIER, J
VALE, W
机构
[1] POPULAT COUNCIL,NEW YORK,NY 10021
[2] SALK INST BIOL STUDIES,PEPTIDE BIOL LAB,LA JOLLA,CA 92037
来源
INTERNATIONAL JOURNAL OF ANDROLOGY | 1982年 / 5卷 / 02期
关键词
D O I
10.1111/j.1365-2605.1982.tb00243.x
中图分类号
R69 [泌尿科学(泌尿生殖系疾病)];
学科分类号
摘要
引用
收藏
页码:158 / 170
页数:13
相关论文
共 32 条
[1]   REDUCTION OF TESTICULAR LUTEINIZING HORMONE HUMAN CHORIONIC-GONADOTROPIN RECEPTORS BY [D-TRP6]-LUTEINIZING HORMONE-RELEASING HORMONE IN HYPOPHYSECTOMIZED RATS [J].
ARIMURA, A ;
SERAFINI, P ;
TALBOT, S ;
SCHALLY, AV .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1979, 90 (03) :687-693
[2]   POTENT INHIBITORY ACTIVITY OF [D-LEU6, DES-GLY-NH210]LHRH ETHYLAMIDE ON LH-HCG AND PRL TESTICULAR RECEPTOR LEVELS IN RAT [J].
AUCLAIR, C ;
KELLY, PA ;
COY, DH ;
SCHALLY, AV ;
LABRIE, F .
ENDOCRINOLOGY, 1977, 101 (06) :1890-1893
[3]   LUTEINIZING-HORMONE-RELEASING HORMONE DOES NOT INHIBIT TESTOSTERONE PRODUCTION IN RAT INTERSTITIAL-CELLS INVITRO [J].
BADGER, TM ;
BEITINS, IZ ;
OSTREA, T ;
CRISAFULLI, JM ;
LITTLE, R ;
SAIDEL, ME .
ENDOCRINOLOGY, 1980, 106 (04) :1149-1153
[4]   EFFECTS OF A LUTEINIZING HORMONE-RELEASING HORMONE ANALOG ON MATING AND FERTILITY IN RATS [J].
BANIK, UK ;
GIVNER, ML .
FERTILITY AND STERILITY, 1976, 27 (09) :1078-1084
[5]   TIME-COURSE OF THE EFFECT OF TREATMENT WITH A POTENT LHRH AGONIST ON TESTICULAR STEROIDOGENESIS AND GONADOTROPIN RECEPTOR LEVELS IN THE ADULT-RAT [J].
BELANGER, A ;
AUCLAIR, C ;
FERLAND, L ;
CARON, S ;
LABRIE, F .
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1980, 13 (02) :191-196
[6]   EFFECTS OF INVIVO ADMINISTRATION OF HUMAN CHORIONIC-GONADOTROPIN AND ETHANOL ON THE PROCESSES OF TESTICULAR RECEPTOR DEPLETION AND REPLENISHMENT [J].
BHALLA, VK ;
CHEN, CJH ;
GNANAPRAKASAM, MS .
LIFE SCIENCES, 1979, 24 (14) :1315-1323
[7]   LUTEINIZING-HORMONE-RELEASING HORMONE-INDUCED REGULATION OF GONADOTROPIN AND PROLACTIN RECEPTORS IN THE RAT TESTIS [J].
CATT, KJ ;
BAUKAL, AJ ;
DAVIES, TF ;
DUFAU, ML .
ENDOCRINOLOGY, 1979, 104 (01) :17-25
[8]   RADIOLIGAND-RECEPTOR ASSAY OF LUTEINIZING-HORMONE AND CHORIONIC GONADOTROPIN [J].
CATT, KJ ;
TSURUHARA, T ;
DUFAU, ML .
JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM, 1972, 34 (01) :123-+
[9]   SPARE GONADOTROPIN RECEPTORS IN RAT TESTIS [J].
CATT, KJ ;
DUFAU, ML .
NATURE-NEW BIOLOGY, 1973, 244 (137) :219-221
[10]   GONADOTROPIN-RELEASING HORMONE ANALOG BINDS TO LUTEAL CELLS AND INHIBITS PROGESTERONE PRODUCTION [J].
CLAYTON, RN ;
HARWOOD, JP ;
CATT, KJ .
NATURE, 1979, 282 (5734) :90-92