A NEW, GENERAL ENTRY TO 4-SUBSTITUTED INDOLES - SYNTHESIS OF (S)-(-)-PINDOLOL AND (+/-)-CHUANGXINMYCIN

被引：33

作者：

ISHIBASHI, H

TABATA, T

HANAOKA, K

IRIYAMA, H

AKAMATSU, S

IKEDA, M

机构：

[1] Kyoto Pharmaceutical University, Kyoto, 607, Misasagi, Yamashina

来源：

TETRAHEDRON LETTERS | 1993年 / 34卷 / 03期

关键词：

D O I：

10.1016/0040-4039(93)85109-A

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A new method for synthesis of 4-substituted indoles has been developed by using the 7-arylthio-6,7-dihydroindol-4(5H)one 5 as a common intermediate. The method was applied to the synthesis of (S)-(-)-pindolol (II) and (+/-)-chuangxinmycin (16).

引用

页码：489 / 492

页数：4

共 16 条

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