INFLUENCE OF SERUM-PROTEIN BINDING ON HEPATIC-CLEARANCE OF S-DISOPYRAMIDE IN THE RABBIT

被引:13
作者
HUANG, JD [1 ]
OIE, S [1 ]
机构
[1] UNIV CALIF SAN FRANCISCO,SCH PHARM,DEPT PHARM,SAN FRANCISCO,CA 94143
关键词
D O I
10.1111/j.2042-7158.1985.tb03042.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:471 / 475
页数:5
相关论文
共 11 条
[1]  
AHMAD AB, 1984, J PHARMACOL EXP THER, V230, P718
[2]  
BALABAUD C, 1973, BIOMED, V23, P353
[3]   RESOLUTION, ABSOLUTE-CONFIGURATION, AND ANTI-ARRHYTHMIC PROPERTIES OF THE ENANTIOMERS OF DISOPYRAMIDE, 4-(DIISOPROPYLAMINO)-2-(2-PYRIDYL)-2-PHENYLBUTYRAMIDE [J].
BURKE, TR ;
NELSON, WL ;
MANGION, M ;
HITE, GJ ;
MOKLER, CM ;
RUENITZ, PC .
JOURNAL OF MEDICINAL CHEMISTRY, 1980, 23 (09) :1044-1048
[4]  
GUENTERT TW, 1980, J PHARMACOL EXP THER, V215, P165
[5]  
HUANG JD, 1983, RES COMMUN CHEM PATH, V41, P227
[6]   HEPATIC ELIMINATION OF DRUGS WITH CONCENTRATION-DEPENDENT SERUM-PROTEIN BINDING [J].
HUANG, JD ;
OIE, S .
JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1984, 12 (01) :67-81
[7]  
Pang K S, 1977, J Pharmacokinet Biopharm, V5, P625, DOI 10.1007/BF01059688
[8]  
PANG KS, 1982, J PHARMACOL EXP THER, V222, P14
[9]   PROTEIN-BINDING AND HEPATIC-CLEARANCE - DISCRIMINATION BETWEEN MODELS OF HEPATIC-CLEARANCE WITH DIAZEPAM, A DRUG OF HIGH INTRINSIC CLEARANCE, IN THE ISOLATED PERFUSED-RAT-LIVER PREPARATION [J].
ROWLAND, M ;
LEITCH, D ;
FLEMING, G ;
SMITH, B .
JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1984, 12 (02) :129-147
[10]   PROTEIN-BINDING AND HEPATIC EXTRACTION OF DIAZEPAM ACROSS THE RAT-LIVER [J].
ROWLAND, M ;
LEITCH, D ;
FLEMING, G ;
SMITH, B .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1983, 35 (06) :383-384