ASYMMETRIC-SYNTHESIS OF CHLORAMPHENICOL

被引：30

作者：

RAO, AVR

RAO, SP

BHANU, MN

机构：

来源：

JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS | 1992年 / 11期

关键词：

D O I：

10.1039/c39920000859

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Enantioselective synthesis of chloramphenicol is described by a route using (2S,3R)-4-nitrophenylglycidol.

引用

页码：859 / 860

页数：2

共 17 条

[1] REGIOSELECTIVE AZIDE OPENING OF 2,3-EPOXY ALCOHOLS BY [TI(O-I-PR)2(N3)2] - SYNTHESIS OF ALPHA-AMINO-ACIDS [J].

CARON, M ;

CARLIER, PR ;

SHARPLESS, KB .

JOURNAL OF ORGANIC CHEMISTRY, 1988, 53 (21) :5185-5187

[2] TI(O-I-PR)4-MEDIATED NUCLEOPHILIC OPENINGS OF 2,3-EPOXY ALCOHOLS - A MILD PROCEDURE FOR REGIOSELECTIVE RING-OPENING [J].

CARON, M ;

SHARPLESS, KB .

JOURNAL OF ORGANIC CHEMISTRY, 1985, 50 (09) :1557-1560

[3] CHLORAMPHENICOL (CHLOROMYCETIN) .5. SYNTHESIS [J].

CONTROULIS, J ;

REBSTOCK, MC ;

CROOKS, HM .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1949, 71 (07) :2463-2468

[4] ALPHA-METHOXY-ALPHA-TRIFLUOROMETHYLPHENYLACETIC ACID, A VERSATILE REAGENT FOR DETERMINATION OF ENANTIOMERIC COMPOSITION OF ALCOHOLS AND AMINES [J].

DALE, JA ;

DULL, DL ;

MOSHER, HS .

JOURNAL OF ORGANIC CHEMISTRY, 1969, 34 (09) :2543-&

[5] AN IMPROVED SYNTHESIS OF THE TAXOL SIDE-CHAIN AND OF RP-56976 [J].

DENIS, JN ;

CORREA, A ;

GREENE, AE .

JOURNAL OF ORGANIC CHEMISTRY, 1990, 55 (06) :1957-1959

[6] CHLOROMYCETIN, A NEW ANTIBIOTIC FROM A SOIL ACTINOMYCETE [J].

EHRLICH, J ;

BARTZ, QR ;

SMITH, RM ;

JOSLYN, DA ;

BURKHOLDER, PR .

SCIENCE, 1947, 106 (2757) :417-417

[7] SELECTIVE TRANSFORMATIONS OF THREO-2,3-DIHYDROXY ESTERS [J].

FLEMING, PR ;

SHARPLESS, KB .

JOURNAL OF ORGANIC CHEMISTRY, 1991, 56 (08) :2869-2875

[8] ANHYDROUS TERT-BUTYL HYDROPEROXIDE IN TOLUENE - THE PREFERRED REAGENT FOR APPLICATIONS REQUIRING DRY TBHP [J].

HILL, JG ;

ROSSITER, BE ;

SHARPLESS, KB .

JOURNAL OF ORGANIC CHEMISTRY, 1983, 48 (20) :3607-3608

[9] SYNTHESIS AND REACTIONS OF 3-HYDROXY-2-NOSYLOXY ESTERS PRODUCED BY THE STEREOSELECTIVE REDUCTION OF 2-NOSYLOXY-3-KETO ESTERS [J].

HOFFMAN, RV ;

KIM, HO .

JOURNAL OF ORGANIC CHEMISTRY, 1991, 56 (24) :6759-6764

[10] ASYMMETRIC DIHYDROXYLATION VIA LIGAND-ACCELERATED CATALYSIS [J].

JACOBSEN, EN ;

MARKO, I ;

MUNGALL, WS ;

SCHRODER, G ;

SHARPLESS, KB .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1988, 110 (06) :1968-1970

← 1 2 →