INHIBITION OF 3(17)BETA-HYDROXYSTEROID DEHYDROGENASE FROM PSEUDOMONAS-TESTOSTERONI BY STEROIDAL A-RING FUSED PYRAZOLES

被引：21

作者：

LEVY, MA

HOLT, DA

BRANDT, M

METCALF, BW

机构：

来源：

BIOCHEMISTRY | 1987年 / 26卷 / 08期

关键词：

D O I：

10.1021/bi00382a030

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：2270 / 2279

页数：10

共 47 条

[1]

ANDERSSON P, 1981, EUR J BIOCH, V113, P549

[2] STRUCTURE OF THE LIVER ALCOHOL DEHYDROGENASE-NAD+-PYRAZOLE COMPLEX AS DETERMINED BY N-15 NMR-SPECTROSCOPY [J].

BECKER, NN ;

ROBERTS, JD .

BIOCHEMISTRY, 1984, 23 (14) :3336-3340

[3]

BIRKTOFT JJ, 1983, J BIOL CHEM, V258, P472

[4] INHIBITION OF TESTOSTERONE 5-ALPHA-REDUCTASE BY A PROPOSED ENZYME-ACTIVATED, ACTIVE SITE-DIRECTED INHIBITOR [J].

BLOHM, TR ;

METCALF, BW ;

LAUGHLIN, ME ;

SJOERDSMA, A ;

SCHATZMAN, GL .

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1980, 95 (01) :273-280

[5]

BRADFORD MM, 1976, ANAL BIOCHEM, V72, P248, DOI 10.1016/0003-2697(76)90527-3

[6] EVIDENCE OF AN ESSENTIAL HISTIDINE RESIDUE IN THERMOLYSIN [J].

BURSTEIN, Y ;

WALSH, KA ;

NEURATH, H .

BIOCHEMISTRY, 1974, 13 (01) :205-210

[7]

Cleland W W, 1979, Methods Enzymol, V63, P103

[8]

Cleland W W, 1977, Adv Enzymol Relat Areas Mol Biol, V45, P273

[9]

CLELAND WW, 1982, METHOD ENZYMOL, V87, P390

[10] STEROIDAL[3,2-C]PYRAZOLES .2. ANDROSTANES, 19-NORANDROSTANES AND THEIR UNSATURATED ANALOGS [J].

CLINTON, RO ;

CHRISTIANSEN, RG ;

CLARKE, RL ;

DEAN, JW ;

MANSON, AJ ;

DICKINSON, WB ;

CARABATEAS, C ;

STONNER, FW ;

ACKERMAN, JH ;

PAGE, DF ;

NEUMANN, HC .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1961, 83 (06) :1478-&

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