GENERATION OF CYTOTOXIC AGENTS BY TARGETED ENZYMES

被引:84
作者
SENTER, PD
WALLACE, PM
SVENSSON, HP
VRUDHULA, VM
KERR, DE
HELLSTROM, I
HELLSTROM, KE
机构
[1] Bristol-Myers Squibb Pharmaceutical Research Institute, Seattle, Washington 98121
关键词
D O I
10.1021/bc00019a001
中图分类号
Q5 [生物化学];
学科分类号
071010 ; 081704 ;
摘要
[No abstract available]
引用
收藏
页码:3 / 9
页数:7
相关论文
共 76 条
[1]   CEPHALOSPORIN NITROGEN-MUSTARD CARBAMATE PRODRUGS FOR ADEPT [J].
ALEXANDER, RP ;
BEELEY, NRA ;
ODRISCOLL, M ;
ONEILL, FP ;
MILLICAN, TA ;
PRATT, AJ ;
WILLENBROCK, FW .
TETRAHEDRON LETTERS, 1991, 32 (27) :3269-3272
[2]   DISPOSITION OF THE PRODRUG 4-(BIS (2-CHLOROETHYL) AMINO) BENZOYL-L-GLUTAMIC ACID AND ITS ACTIVE PARENT DRUG IN MICE [J].
ANTONIW, P ;
SPRINGER, CJ ;
BAGSHAWE, KD ;
SEARLE, F ;
MELTON, RG ;
ROGERS, GT ;
BURKE, PJ ;
SHERWOOD, RF .
BRITISH JOURNAL OF CANCER, 1990, 62 (06) :909-914
[3]  
BAGSHAWE KD, 1991, ANTIBODY IMMUNOCONJ, V4, P915
[4]   A CYTO-TOXIC AGENT CAN BE GENERATED SELECTIVELY AT CANCER SITES [J].
BAGSHAWE, KD ;
SPRINGER, CJ ;
SEARLE, F ;
ANTONIW, P ;
SHARMA, SK ;
MELTON, RG ;
SHERWOOD, RF .
BRITISH JOURNAL OF CANCER, 1988, 58 (06) :700-703
[5]   ISOLATION OF HIGHLY MALIGNANT THY-1-POSITIVE REVERTANTS FROM CULTURED CLONED THY-1-NEGATIVE LYMPHOMA-CELLS OF LOW TUMORIGENICITY [J].
BASCH, RS ;
LAKOW, E ;
TENG, M ;
BUXBAUM, JN .
SOMATIC CELL AND MOLECULAR GENETICS, 1984, 10 (01) :37-44
[6]  
BATTELLI MG, 1988, CLIN EXP IMMUNOL, V73, P128
[7]  
BIGNAMI GS, 1992, IN PRESS CANCER RES
[8]   ROLES OF UDP-GLUCURONOSYLTRANSFERASES IN CHEMICAL CARCINOGENESIS [J].
BOCK, KW .
CRITICAL REVIEWS IN BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1991, 26 (02) :129-150
[9]   MOLECULAR AND FUNCTIONAL-CHARACTERIZATION OF A FUSION PROTEIN SUITED FOR TUMOR SPECIFIC PRODRUG ACTIVATION [J].
BOSSLET, K ;
CZECH, J ;
LORENZ, P ;
SEDLACEK, HH ;
SCHUERMANN, M ;
SEEMANN, G .
BRITISH JOURNAL OF CANCER, 1992, 65 (02) :234-238
[10]   A BRIEF SURVEY OF METHODS FOR PREPARING PROTEIN CONJUGATES WITH DYES, HAPTENS, AND CROSS-LINKING REAGENTS [J].
BRINKLEY, M .
BIOCONJUGATE CHEMISTRY, 1992, 3 (01) :2-13