TISSUE AND SUBSTRATE-SPECIFICITY OF INHIBITION BY ALKOXY-ARYL-LACTAMS OF PLATELET AND ARTERIAL SMOOTH-MUSCLE CYCLIC-NUCLEOTIDE PHOSPHODIESTERASES RELATIONSHIP TO PHARMACOLOGICAL ACTIVITY

被引：63

作者：

LUGNIER, C

STIERLE, A

BERETZ, A

SCHOEFFTER, P

LEBEC, A

WERMUTH, CG

CAZENAVE, JP

STOCLET, JC

机构：

[1] FAC PHARM STRASBOURG,INSERM,U243,F-67048 STRASBOURG,FRANCE

[2] FAC PHARM STRASBOURG,CHIM ORGAN LAB,CNRS,ERA 393,F-67048 STRASBOURG,FRANCE

[3] CTR TRANSFUS SANGUINE,BIOL & PHARMACOL PLAQUETTES LAB,F-67085 STRASBOURG,FRANCE

来源：

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS | 1983年 / 113卷 / 03期

关键词：

D O I：

10.1016/0006-291X(83)91091-4

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：954 / 959

页数：6

共 18 条

[1] IDENTIFICATION AND PROPERTIES OF CYCLIC-NUCLEOTIDE PHOSPHODIESTERASES [J].

BEAVO, JA ;

HANSEN, RS ;

HARRISON, SA ;

HURWITZ, RL ;

MARTINS, TJ ;

MUMBY, MC .

MOLECULAR AND CELLULAR ENDOCRINOLOGY, 1982, 28 (03) :387-410

[2] INHIBITION OF AGGREGATION AND SECRETION OF HUMAN-PLATELETS BY QUERCETIN AND OTHER FLAVONOIDS - STRUCTURE ACTIVITY RELATIONSHIPS [J].

BERETZ, A ;

CAZENAVE, JP ;

ANTON, R .

AGENTS AND ACTIONS, 1982, 12 (03) :382-387

[3] INHIBITION OF CYCLIC-AMP PHOSPHODIESTERASE ACTIVITY AND MYOCARDIAL-CONTRACTILITY - EFFECTS OF CILOSTAMIDE, A NOVEL PDE INHIBITOR, AND METHYLISOBUTYLXANTHINE ON RABBIT AND CANINE VENTRICULAR MUSCLE [J].

ENDOH, M ;

SATOH, K ;

YAMASHITA, S .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1980, 66 (01) :43-52

[4]

FURCHGOTT RF, 1953, J PHARMACOL EXP THER, V108, P129

[5] HUMAN-BLOOD PLATELET 3' - 5'-CYCLIC NUCLEOTIDE PHOSPHODIESTERASE - ISOLATION OF LOW-KM AND HIGH-KM PHOSPHODIESTERASE [J].

HIDAKA, H ;

ASANO, T .

BIOCHIMICA ET BIOPHYSICA ACTA, 1976, 429 (02) :485-497

[6]

HIDAKA H, 1979, J PHARMACOL EXP THER, V211, P26

[7] CYCLIC-NUCLEOTIDE PHOSPHODIESTERASE ACTIVITIES FROM PIG CORONARY-ARTERIES - LACK OF INTERCONVERTIBILITY OF MAJOR FORMS [J].

KERAVIS, TM ;

WELLS, JN ;

HARDMAN, JG .

BIOCHIMICA ET BIOPHYSICA ACTA, 1980, 613 (01) :116-129

[8]

KINLOUGHRATHBONE RL, 1977, THROMB HAEMOSTASIS, V37, P291

[9] SELECTIVE-INHIBITION OF CYCLIC NUCLEOTIDE PHOSPHODIESTERASES BY ANALOGS OF 1-METHYL-3-ISOBUTYLXANTHINE [J].

KRAMER, GL ;

GARST, JE ;

MITCHEL, SS ;

WELLS, JN .

BIOCHEMISTRY, 1977, 16 (15) :3316-3321

[10] CYCLIC NUCLEOTIDE PHOSPHODIESTERASE INHIBITION AND VASCULAR SMOOTH MUSCLE RELAXATION [J].

LUGNIER, C ;

BERTRAND, Y ;

STOCLET, JC .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1972, 19 (01) :134-&

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