INCREASED ANALGESIC POTENCY OF MORPHINE AND INCREASED BRAIN OPIOID BINDING-SITES IN THE RAT FOLLOWING CHRONIC NALTREXONE TREATMENT

被引:82
作者
YOBURN, BC [1 ]
GOODMAN, RR [1 ]
COHEN, AH [1 ]
PASTERNAK, GW [1 ]
INTURRISI, CE [1 ]
机构
[1] MEM SLOAN KETTERING CANC CTR,COTZIAS LAB NEUROONCOL,NEW YORK,NY 10021
关键词
D O I
10.1016/0024-3205(85)90322-4
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
引用
收藏
页码:2325 / 2332
页数:8
相关论文
共 31 条
[1]   AGE-RELATED DIFFERENCES IN THE EFFECT OF CHRONIC ADMINISTRATION OF NALOXONE ON OPIATE BINDING IN RAT-BRAIN [J].
BARDO, MT ;
BHATNAGAR, RK ;
GEBHART, GF .
NEUROPHARMACOLOGY, 1983, 22 (04) :453-461
[2]   CHRONIC NALTREXONE INCREASES OPIATE BINDING IN BRAIN AND PRODUCES SUPERSENSITIVITY TO MORPHINE IN THE LOCUS COERULEUS OF THE RAT [J].
BARDO, MT ;
BHATNAGAR, RK ;
GEBHART, GF .
BRAIN RESEARCH, 1983, 289 (1-2) :223-234
[3]   DIFFERENTIAL-EFFECTS OF CHRONIC MORPHINE AND NALOXONE ON OPIATE RECEPTORS, MONOAMINES, AND MORPHINE-INDUCED BEHAVIORS IN PREWEANLING RATS [J].
BARDO, MT ;
BHATNAGAR, RK ;
GEBHART, GF .
DEVELOPMENTAL BRAIN RESEARCH, 1982, 4 (02) :139-147
[4]   MODULATION OF OPIOID SYSTEM IN C57 MICE AFTER REPEATED TREATMENT WITH MORPHINE AND NALOXONE - BIOCHEMICAL AND BEHAVIORAL-CORRELATES [J].
BRUNELLO, N ;
VOLTERRA, A ;
DIGIULIO, AM ;
CUOMO, V ;
RACAGNI, G .
LIFE SCIENCES, 1984, 34 (17) :1669-1678
[5]  
CHANG KJ, 1979, J BIOL CHEM, V254, P2610
[6]   OPIOID-PEPTIDES INDUCE REDUCTION OF ENKEPHALIN RECEPTORS IN CULTURED NEURO-BLASTOMA CELLS [J].
CHANG, KJ ;
ECKEL, RW ;
BLANCHARD, SG .
NATURE, 1982, 296 (5856) :446-448
[7]  
DAVIS ME, 1979, J PHARMACOL EXP THER, V211, P112
[8]  
Finney D. J., 1971, PROBIT ANAL
[9]   NALOXONE RADIOIMMUNOASSAY - AN IMPROVED ANTI-SERUM [J].
HAHN, EF ;
LAHITA, R ;
KREEK, MJ ;
DUMA, C ;
INTURRISI, CE .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1983, 35 (12) :833-836
[10]   NALOXAZONE IRREVERSIBLY INHIBITS THE HIGH-AFFINITY BINDING OF [I-125]D-ALA2-D-LEU5-ENKEPHALIN [J].
HAZUM, E ;
CHANG, KJ ;
CUATRECASAS, P ;
PASTERNAK, GW .
LIFE SCIENCES, 1981, 28 (26) :2973-2979