MECHANISM-BASED INACTIVATION OF N-ARYLHYDROXAMIC ACID N,O-ACYLTRANSFERASE BY 7-SUBSTITUTED-N-HYDROXY-2-ACETAMIDOFLUORENES

被引：27

作者：

MARHEVKA, VC

EBNER, NA

SEHON, RD

HANNA, PE

机构：

[1] UNIV MINNESOTA,DEPT MED CHEM,MINNEAPOLIS,MN 55455

[2] UNIV MINNESOTA,DEPT PHARMACOL,MINNEAPOLIS,MN 55455

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1985年 / 28卷 / 01期

关键词：

D O I：

10.1021/jm00379a005

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：18 / 24

页数：7

共 34 条

[1] NITRATION OF 3-METHOXYFLUORANTHENE [J].

ANDREW, HF ;

CAMPBELL, N ;

CRAIG, JT ;

NICHOL, KJ .

JOURNAL OF THE CHEMICAL SOCIETY C-ORGANIC, 1968, (14) :1761-&

[2] ELECTROPHILIC N-ACETOXYAMINOARENES DERIVED FROM CARCINOGENIC N-HYDROXY-N-ACETYLAMINOARENES BY ENZYMATIC DEACETYLATION AND TRANSACETYLATION IN LIVER [J].

BARTSCH, H ;

DWORKIN, M ;

MILLER, JA ;

MILLER, EC .

BIOCHIMICA ET BIOPHYSICA ACTA, 1972, 286 (02) :272-298

[3] ACETYL TRANSFER IN ARYLAMINE METABOLISM [J].

BOOTH, J .

BIOCHEMICAL JOURNAL, 1966, 100 (03) :745-&

[4] COMPARISON OF THE INHIBITION OF METHOTREXATE-SENSITIVE AND METHOTREXATE-RESISTANT LACTOBACILLUS-CASEI CELL-CULTURES WITH PURIFIED LACTOBACILLUS-CASEI DIHYDROFOLATE-REDUCTASE BY 4,6-DIAMINO-1,2-DIHYDRO-2,2-DIMETHYL-1-(3-SUBSTITUTED-PHENYL)-S-TRIAZINES - USE OF QUANTITATIVE STRUCTURE-ACTIVITY-RELATIONSHIPS IN MAKING INFERENCES ABOUT THE MECHANISM OF RESISTANCE AND THE STRUCTURE OF THE ENZYME INSITU COMPARED WITH THE ENZYME INVITROUA [J].

COATS, EA ;

GENTHER, CS ;

DIETRICH, SW ;

GUO, Z ;

HANSCH, C .

JOURNAL OF MEDICINAL CHEMISTRY, 1981, 24 (12) :1422-1429

[5] FREE-RADICAL EVENTS IN CHEMICAL AND BIOCHEMICAL REACTIONS INVOLVING CARCINOGENIC ARYLAMINES [J].

FLOYD, RA .

RADIATION RESEARCH, 1981, 86 (02) :243-263

[6] MNDO MOLECULAR-ORBITAL STUDY OF NITRENIUM IONS DERIVED FROM CARCINOGENIC AROMATIC-AMINES AND AMIDES [J].

FORD, GP ;

SCRIBNER, JD .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1981, 103 (15) :4281-4291

[7] REACTIONS OF PER ACIDS .1. THE REACTION OF PERBENZOIC ACID WITH SOME SIMPLE KETONES [J].

FRIESS, SL .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1949, 71 (01) :14-15

[8] SYNTHESIS AND REARRANGEMENT OF METHANESULFONATE ESTERS OF N-HYDROXYACETANILIDES - A MODEL FOR A PENULTIMATE CARCINOGEN [J].

GASSMAN, PG ;

GRANRUD, JE .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1984, 106 (05) :1498-1499

[9]

GLOWINSKI IB, 1980, J BIOL CHEM, V255, P7883

[10] A NEW SYNTHESIS OF 2-CHLORO-7-NITROFLUORENE [J].

GUTMANN, HR ;

RAY, FE .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1951, 73 (08) :4033-4033

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