HUMAN PROGESTERONE-RECEPTOR COMPLEXED WITH THE ANTAGONIST RU-486 BINDS TO HORMONE RESPONSE ELEMENTS IN A STRUCTURALLY ALTERED FORM

被引:133
作者
ELASHRY, D [1 ]
ONATE, SA [1 ]
NORDEEN, SK [1 ]
EDWARDS, DP [1 ]
机构
[1] UNIV COLORADO,HLTH SCI CTR,DEPT PATHOL B216,4200 E 9TH ST,DENVER,CO 80262
关键词
D O I
10.1210/mend-3-10-1545
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:1545 / 1558
页数:14
相关论文
共 34 条
[1]   ACTIVATION OF RAT-LIVER GLUCOCORTICOID RECEPTOR BOUND TO THE ANTIGLUCOCORTICOID RU38486 [J].
AGARWAL, MK ;
LOMBARDO, G ;
ELIEZER, N ;
MOUDGIL, VK .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1985, 133 (02) :745-752
[2]   STEROID HORMONE-DEPENDENT INTERACTION OF HUMAN PROGESTERONE-RECEPTOR WITH ITS TARGET ENHANCER ELEMENT [J].
BAGCHI, MK ;
ELLISTON, JF ;
TSAI, SY ;
EDWARDS, DP ;
TSAI, MJ ;
OMALLEY, BW .
MOLECULAR ENDOCRINOLOGY, 1988, 2 (12) :1221-1229
[3]   SEQUENCE-SPECIFIC DNA-BINDING OF THE PROGESTERONE-RECEPTOR TO THE UTEROGLOBIN GENE - EFFECTS OF HORMONE, ANTIHORMONE AND RECEPTOR PHOSPHORYLATION [J].
BAILLY, A ;
LEPAGE, C ;
RAUCH, M ;
MILGROM, E .
EMBO JOURNAL, 1986, 5 (12) :3235-3241
[4]   STEROID-HORMONE ANTAGONISTS AT THE RECEPTOR LEVEL - A ROLE FOR THE HEAT-SHOCK PROTEIN MW 90,000 (HSP-90) [J].
BAULIEU, EE .
JOURNAL OF CELLULAR BIOCHEMISTRY, 1987, 35 (02) :161-174
[5]   DNA-BINDING PROPERTIES OF GLUCOCORTICOSTEROID RECEPTORS BOUND TO THE STEROID ANTAGONIST RU-486 [J].
BOURGEOIS, S ;
PFAHL, M ;
BAULIEU, EE .
EMBO JOURNAL, 1984, 3 (04) :751-755
[6]   REQUIREMENT OF HORMONE FOR THERMAL-CONVERSION OF THE GLUCOCORTICOID RECEPTOR TO A DNA-BINDING STATE [J].
DENIS, M ;
POELLINGER, L ;
WIKSTOM, AC ;
GUSTAFSSON, JA .
NATURE, 1988, 333 (6174) :686-688
[7]   HUMAN PROGESTERONE-RECEPTOR BINDING TO MOUSE MAMMARY-TUMOR VIRUS DEOXYRIBONUCLEIC-ACID - DEPENDENCE ON HORMONE AND NONRECEPTOR NUCLEAR FACTOR(S) [J].
EDWARDS, DP ;
KUHNEL, B ;
ESTES, PA ;
NORDEEN, SK .
MOLECULAR ENDOCRINOLOGY, 1989, 3 (02) :381-391
[8]  
ELASHRYSTOWERS D, 1988, CANCER RS, V48, P6464
[9]   IMMUNOLOGICAL ANALYSIS OF HUMAN-BREAST CANCER PROGESTERONE RECEPTORS .1. IMMUNOAFFINITY PURIFICATION OF TRANSFORMED RECEPTORS AND PRODUCTION OF MONOCLONAL-ANTIBODIES [J].
ESTES, PA ;
SUBA, EJ ;
LAWLERHEAVNER, J ;
ELASHRYSTOWERS, D ;
WEI, LL ;
TOFT, DO ;
SULLIVAN, WP ;
HORWITZ, KB ;
EDWARDS, DP .
BIOCHEMISTRY, 1987, 26 (19) :6250-6262
[10]   ANTIGLUCOCORTICOSTEROID EFFECTS SUGGEST WHY STEROID-HORMONE IS REQUIRED FOR RECEPTORS TO BIND DNA INVIVO BUT NOT INVITRO [J].
GROYER, A ;
SCHWEIZERGROYER, G ;
CADEPOND, F ;
MARILLER, M ;
BAULIEU, EE .
NATURE, 1987, 328 (6131) :624-626