MODIFICATION OF PYRAZOLOQUINOLINONE AFFINITY BY GABA PREDICTS EFFICACY AT THE BENZODIAZEPINE RECEPTOR

被引:7
作者
BROWN, CL
MARTIN, IL
机构
关键词
D O I
10.1016/0014-2999(84)90691-5
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:167 / 173
页数:7
相关论文
共 16 条
[1]   INTERACTION OF CONVULSIVE LIGANDS WITH BENZODIAZEPINE RECEPTORS [J].
BRAESTRUP, C ;
SCHMIECHEN, R ;
NEEF, G ;
NIELSEN, M ;
PETERSEN, EN .
SCIENCE, 1982, 216 (4551) :1241-1243
[2]   GABA REDUCES BINDING OF H-3-LABELED METHYL BETA-CARBOLINE-3-CARBOXYLATE TO BRAIN BENZODIAZEPINE RECEPTORS [J].
BRAESTRUP, C ;
NIELSEN, M .
NATURE, 1981, 294 (5840) :472-474
[3]   INVIVO DETERMINATION OF EFFICACY OF PYRAZOLOQUINOLINONES AT THE BENZODIAZEPINE RECEPTOR [J].
BROWN, C ;
MARTIN, I ;
JONES, B ;
OAKLEY, N .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 103 (1-2) :139-143
[4]  
DOBLE A, 1982, British Journal of Pharmacology, V76, p238P
[5]   ENDOGENOUS PROTEIN MODULATES AFFINITY OF GABA AND BENZODIAZEPINE RECEPTORS IN RAT-BRAIN [J].
GUIDOTTI, A ;
TOFFANO, G ;
COSTA, E .
NATURE, 1978, 275 (5680) :553-555
[6]   CENTRAL ACTIONS OF BENZODIAZEPINES - GENERAL INTRODUCTION [J].
HAEFELY, WE .
BRITISH JOURNAL OF PSYCHIATRY, 1978, 133 (SEP) :231-238
[7]   SELECTIVE ANTAGONISTS OF BENZODIAZEPINES [J].
HUNKELER, W ;
MOHLER, H ;
PIERI, L ;
POLC, P ;
BONETTI, EP ;
CUMIN, R ;
SCHAFFNER, R ;
HAEFELY, W .
NATURE, 1981, 290 (5806) :514-516
[8]  
KEIM KL, 1984, FED PROC, V43, P930
[9]   AGONIST AND ANTAGONIST BENZODIAZEPINE RECEPTOR INTERACTION INVITRO [J].
MOHLER, H ;
RICHARDS, JG .
NATURE, 1981, 294 (5843) :763-765
[10]   BENZODIAZEPINE RECEPTOR - DEMONSTRATION IN CENTRAL NERVOUS-SYSTEM [J].
MOHLER, H ;
OKADA, T .
SCIENCE, 1977, 198 (4319) :849-851