NMDA RECEPTOR ANTAGONISTS THAT BIND TO THE STRYCHNINE-INSENSITIVE GLYCINE SITE AND INHIBIT NMDA-INDUCED CA-2+ FLUXES AND [H-3]GABA RELEASE

被引：48

作者：

REYNOLDS, IJ ^{[1
]}

HARRIS, KM ^{[1
]}

MILLER, RJ ^{[1
]}

机构：

[1] UNIV CHICAGO,DEPT PHARMACOL & PHYSIOL SCI,947 E 58TH ST,CHICAGO,IL 60637

来源：

EUROPEAN JOURNAL OF PHARMACOLOGY-MOLECULAR PHARMACOLOGY SECTION | 1989年 / 172卷 / 01期

关键词：

D O I：

10.1016/0922-4106(89)90040-0

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

引用

页码：9 / 17

页数：9

共 27 条

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[3] GLYCINE REVERSES ANTAGONISM OF N-METHYL-D-ASPARTATE (NMDA) BY 1-HYDROXY-3-AMINOPYRROLIDONE-2 (HA-966) BUT NOT BY D-2-AMINO-5-PHOPHONOVALERATE (D-AP5) ON RAT CORTICAL SLICES [J].

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EUROPEAN JOURNAL OF PHARMACOLOGY, 1988, 151 (01) :161-162

[4] THE NOVEL ANTICONVULSANT MK-801 BINDS TO THE ACTIVATED STATE OF THE N-METHYL-D-ASPARTATE RECEPTOR IN RAT-BRAIN [J].

FOSTER, AC ;

WONG, EHF .

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[5]

HARRIS KM, IN PRESS BRAIN RES

[6] KETAMINE AND PHENCYCLIDINE CAUSE A VOLTAGE-DEPENDENT BLOCK OF RESPONSES TO L-ASPARTIC ACID [J].

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MILJKOVIC, Z ;

MACDONALD, JF .

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[7] BLOCK OF N-METHYL-D-ASPARTATE-ACTIVATED CURRENT BY THE ANTICONVULSANT MK-801 - SELECTIVE BINDING TO OPEN CHANNELS [J].

HUETTNER, JE ;

BEAN, BP .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1988, 85 (04) :1307-1311

[8] GLYCINE POTENTIATES THE NMDA RESPONSE IN CULTURED MOUSE-BRAIN NEURONS [J].

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ASCHER, P .

NATURE, 1987, 325 (6104) :529-531

[9] NONCOMPETITIVE ANTAGONISTS OF EXCITATORY AMINO-ACID RECEPTORS [J].

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FOSTER, AC ;

WONG, EHF .

TRENDS IN NEUROSCIENCES, 1987, 10 (07) :294-298

[10] 7-CHLOROKYNURENIC ACID IS A SELECTIVE ANTAGONIST AT THE GLYCINE MODULATORY SITE OF THE N-METHYL-D-ASPARTATE RECEPTOR COMPLEX [J].

KEMP, JA ;

FOSTER, AC ;

LEESON, PD ;

PRIESTLEY, T ;

TRIDGETT, R ;

IVERSEN, LL ;

WOODRUFF, GN .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1988, 85 (17) :6547-6550

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