GAMMA-AMINOBUTYRIC ACID MODULATION OF BENZODIAZEPINE RECEPTOR-BINDING INVITRO DOES NOT PREDICT THE PHARMACOLOGIC ACTIVITY OF ALL BENZODIAZEPINE RECEPTOR LIGANDS

被引:7
作者
CHWEH, AY
SWINYARD, EA
WOLF, HH
机构
关键词
D O I
10.1016/S0304-3940(85)80074-4
中图分类号
Q189 [神经科学];
学科分类号
071006 ;
摘要
引用
收藏
页码:173 / 177
页数:5
相关论文
共 18 条
[1]   BENZODIAZEPINE RECEPTOR LIGANDS WITH POSITIVE AND NEGATIVE EFFICACY [J].
BRAESTRUP, C ;
NIELSEN, M ;
HONORE, T ;
JENSEN, LH ;
PETERSEN, EN .
NEUROPHARMACOLOGY, 1983, 22 (12B) :1451-1457
[2]   EFFECT OF GABA AGONISTS ON THE NEUROTOXICITY AND ANTICONVULSANT ACTIVITY OF BENZODIAZEPINES [J].
CHWEH, AY ;
SWINYARD, EA ;
WOLF, HH ;
KUPFERBERG, HJ .
LIFE SCIENCES, 1985, 36 (08) :737-744
[3]   HYPNOTIC ACTION OF BENZODIAZEPINES - A POSSIBLE MECHANISM [J].
CHWEH, AY ;
LIN, YB ;
SWINYARD, EA .
LIFE SCIENCES, 1984, 34 (18) :1763-1768
[4]  
DOBLE A, 1982, British Journal of Pharmacology, V76, p238P
[5]   MODULATION OF BENZODIAZEPINE RECEPTOR-BINDING - INSIGHT INTO PHARMACOLOGICAL EFFICACY [J].
EHLERT, FJ ;
RAGAN, P ;
CHEN, A ;
ROESKE, WR ;
YAMAMURA, HI .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1982, 78 (02) :249-253
[6]  
Finney DJ, 1971, PROBIT ANAL, V3rd, P81
[7]  
MARANGOS PJ, 1981, MOL PHARMACOL, V20, P16
[8]   AGONIST AND ANTAGONIST BENZODIAZEPINE RECEPTOR INTERACTION INVITRO [J].
MOHLER, H ;
RICHARDS, JG .
NATURE, 1981, 294 (5843) :763-765
[9]   NICOTINAMIDE IS A BRAIN CONSTITUENT WITH BENZODIAZEPINE-LIKE ACTIONS [J].
MOHLER, H ;
POLC, P ;
CUMIN, R ;
PIERI, L ;
KETTLER, R .
NATURE, 1979, 278 (5704) :563-565
[10]   PROPERTIES OF DIAZEPAM-H-3 BINDING TO BENZODIAZEPINE RECEPTORS IN RAT CEREBRAL-CORTEX [J].
MOHLER, H ;
OKADA, T .
LIFE SCIENCES, 1977, 20 (12) :2101-2110