QUANTITATIVE RELATIONSHIPS BETWEEN ALPHA-ADRENERGIC ACTIVITY AND BINDING-AFFINITY OF ALPHA-ADRENOCEPTOR AGONISTS AND ANTAGONISTS

被引：35

作者：

TIMMERMANS, PBMWM

DEJONGE, A

THOOLEN, MJMC

WILFFERT, B

BATINK, H

VANZWIETEN, PA

机构：

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1984年 / 27卷 / 04期

关键词：

D O I：

10.1021/jm00370a011

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：495 / 503

页数：9

共 75 条

[1]

Ariens EJ, 1964, MOL PHARM, V2

[2] SOME QUANTITATIVE USES OF DRUG ANTAGONISTS [J].

ARUNLAKSHANA, O ;

SCHILD, HO .

BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1959, 14 (01) :48-58

[3]

BERLAN M, 1982, J PHYSIOLOGY PARIS, V78, P279

[4] FUNCTIONAL BASIS FOR CLASSIFICATION OF ALPHA-ADRENERGIC RECEPTORS [J].

BERTHELSEN, S ;

PETTINGER, WA .

LIFE SCIENCES, 1977, 21 (05) :595-606

[5] COMPARISON OF PRESYNAPTIC AND POSTSYNAPTIC EFFECTS OF ALPHA-ADRENOLYTIC DRUGS IN PULMONARY-ARTERY OF RABBIT [J].

BOROWSKI, E ;

STARKE, K ;

EHRL, H ;

ENDO, T .

NEUROSCIENCE, 1977, 2 (02) :285-296

[6] [H-3]-LABELED RAUWOLSCINE AND [H-3]-LABELED YOHIMBINE BINDING TO RAT CEREBRAL AND HUMAN-PLATELET MEMBRANES - POSSIBLE HETEROGENEITY OF ALPHA-2-ADRENOCEPTORS [J].

CHEUNG, YD ;

BARNETT, DB ;

NAHORSKI, SR .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1982, 84 (1-2) :79-85

[7] HUMAN-PLATELET ALPHA-2-ADRENERGIC RECEPTORS - LABELING WITH YOHIMBINE-H-3, A SELECTIVE ANTAGONIST LIGAND [J].

DAIGUJI, M ;

MELTZER, HY ;

UPRICHARD, DC .

LIFE SCIENCES, 1981, 28 (24) :2705-2717

[8]

DEJONG AP, 1981, EUR J PHARMACOL, V69, P175

[9]

DEJONGE A, 1983, J PHARMACOL EXP THER, V226, P565

[10]

DEJONGE A, 1981, J AUTON PHARMACOL, V1, P377

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