学术探索
学术期刊
新闻热点
数据分析
智能评审

QUANTITATIVE RELATIONSHIPS BETWEEN ALPHA-ADRENERGIC ACTIVITY AND BINDING-AFFINITY OF ALPHA-ADRENOCEPTOR AGONISTS AND ANTAGONISTS

被引：35
作者：
TIMMERMANS, PBMWM
DEJONGE, A
THOOLEN, MJMC
WILFFERT, B
BATINK, H
VANZWIETEN, PA
机构：
来源：
JOURNAL OF MEDICINAL CHEMISTRY | 1984年 / 27卷 / 04期
关键词：
D O I：
10.1021/jm00370a011
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
引用
收藏
页码：495 / 503
页数：9
相关论文
共 75 条
[51]   RELATIVE PRESYNAPTIC AND POSTSYNAPTIC POTENCIES OF ALPHA-ADRENOCEPTOR AGONISTS IN RABBIT PULMONARY-ARTERY [J].
STARKE, K ;
ENDO, T ;
TAUBE, HD .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1975, 291 (01) :55-78
[52]   MODIFICATION OF RECEPTOR THEORY [J].
STEPHENSON, RP .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1956, 11 (04) :379-393
[53]   DISPLACEMENT OF [CLONIDINE-H-3 BINDING BY CLONIDINE ANALOGS IN MEMBRANES FROM RAT CEREBRAL-CORTEX [J].
SUMMERS, RJ ;
JARROTT, B ;
LOUIS, WJ .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1980, 66 (2-3) :233-241
[54]   BINDING OF H-3-CLONIDINE TO AN ALPHA-ADRENOCEPTOR IN MEMBRANES OF GUINEA-PIG ILEUM [J].
TANAKA, T ;
STARKE, K .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1979, 309 (03) :207-215
[55]   CHARACTERIZATION OF ALPHA-ADRENOCEPTOR POPULATIONS - QUANTITATIVE RELATIONSHIPS BETWEEN CARDIOVASCULAR EFFECTS INITIATED AT CENTRAL AND PERIPHERAL ALPHA-ADRENOCEPTORS [J].
TIMMERMANS, PBMWM ;
DEJONGE, A ;
VANMEEL, JCA ;
SLOTHORSTGRISDIJK, FP ;
LAM, E ;
VANZWIETEN, PA .
JOURNAL OF MEDICINAL CHEMISTRY, 1981, 24 (05) :502-507
[56]   ALPHA-1/ALPHA-2-ADRENOCEPTOR AGONIST SELECTIVITY OF MONO AND DIHYDROXY-2-N,N-DI-NORMAL-PROPYLAMINOTETRALINS [J].
TIMMERMANS, PBMWM ;
MATHY, MJ ;
WILFFERT, B ;
KALKMAN, HO ;
SMIT, G ;
DIJKSTRA, D ;
HORN, AS ;
VANZWIETEN, PA .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 97 (1-2) :55-65
[57]  
TIMMERMANS PBMWM, 1981, MOL PHARMACOL, V20, P295
[58]   CHARACTERIZATION OF ALPHA-ADRENOCEPTORS PARTICIPATING IN THE CENTRAL HYPOTENSIVE AND SEDATIVE EFFECTS OF CLONIDINE USING YOHIMBINE, RAUWOLSCINE AND CORYNANTHINE [J].
TIMMERMANS, PBMWM ;
SCHOOP, AMC ;
KWA, HY ;
VANZWIETEN, HA .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1981, 70 (01) :7-15
[59]   VASOCONSTRICTION MEDIATED BY POSTSYNAPTIC ALPHA-2-ADRENOCEPTOR STIMULATION [J].
TIMMERMANS, PBMWM ;
VANZWIETEN, PA .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1980, 313 (01) :17-20
[60]   SELECTIVITY OF BENZODIOXANE ALPHA-ADRENOCEPTOR ANTAGONISTS FOR ALPHA-1-ADRENOCEPTORS AND ALPHA-2-ADRENOCEPTOR DETERMINED BY BINDING-AFFINITY [J].
TIMMERMANS, PBMWM ;
VANKEMENADE, JE ;
BATINK, HD ;
VANZWIETEN, PA .
PHARMACOLOGY, 1983, 26 (05) :258-269
12345678