INTRAMOLECULAR ALKYLATION OF CARBOXYLIC-ACIDS - APPLICATION TO THE SYNTHESIS OF BOC-PROTECTED CYCLIC AMINO-ACIDS

被引：14

作者：

DENICOLA, A

EINHORN, C

EINHORN, J

LUCHE, JL

机构：

[1] UNIV J FOURIER,ETUD DYNAM & STRUCT SELECTIV LAB,BATIMENT CHIM,BP 53X,F-38041 GRENOBLE,FRANCE

[2] UNIV TOULOUSE 3,LAB AMPERES,CNRS,EP 52,F-31062 TOULOUSE,FRANCE

来源：

JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS | 1994年 / 07期

关键词：

D O I：

10.1039/c39940000879

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

A new synthesis of Boc-protected cyclic amino acids is described as an application of an unreported method of lithium diisopropylamide-induced cyclisation of omega-chloro carboxylic acids containing a protected amine function in the chain.

引用

页码：879 / 880

页数：2

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