INVITRO INHIBITION OF ESTROGEN SULFOCONJUGATION BY SOME 2-SUBSTITUTED AND 4-SUBSTITUTED "ESTRA-1,3,5(10)-TRIEN-17-BETA-OLS1A

被引：21

作者：

HORWITZ, JP

IYER, VK

VARDHAN, HB

COROMBOS, J

BROOKS, SC

机构：

[1] WAYNE STATE UNIV,SCH MED,DEPT BIOCHEM,DETROIT,MI 48201

[2] WAYNE STATE UNIV,SCH MED,DEPT MED,DETROIT,MI 48201

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1986年 / 29卷 / 05期

关键词：

D O I：

10.1021/jm00155a019

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：692 / 698

页数：7

共 40 条

[21] REPLACEMENT OF PHENOLIC HYDROXYL GROUPS BY HYDROGEN [J].

MUSLINER, WJ ;

GATES, JW .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1966, 88 (18) :4271-&

[22]

NAMBARA T, 1971, CHEM PHARM BULL, V19, P153

[23] REGIOSPECIFIC SYNTHESES OF MODIFIED STEROID-HORMONES .2. 4-FLUORO-17-ESTRADIOL AND 4-FLUORO-17BETA-ESTRONE [J].

NEEMAN, M ;

OSAWA, Y ;

MUKAI, T .

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 1972, (18) :2297-&

[24]

NEEMAN R, 1963, TETRAHEDRON LETT, P1987

[25] SYNTHESIS OF 4-FLUOROESTRADIOL ANALOGS [J].

NJAR, VCO ;

ARUNACHALAM, T ;

CASPI, E .

JOURNAL OF ORGANIC CHEMISTRY, 1983, 48 (07) :1007-1011

[26] CYCLIC ACTIVITY OF ESTROGEN SULFOTRANSFERASE IN GILT UTERUS [J].

PACK, BA ;

BROOKS, SC .

ENDOCRINOLOGY, 1974, 95 (06) :1680-1690

[27]

PACK BA, 1974, J CLIN ENDOCRINOL ME, V48, P420

[28]

PEWNIM T, 1980, CANCER RES, V40, P1360

[29]

ROE A, 1949, ORGANIC REACTIONS, V5, pCH4

[30] SODIUM-BOROHYDRIDE REDUCTIONS UNDER PHASE-TRANSFER CONDITIONS - CONVERSION OF HALIDES AND SULFONATE ESTERS TO ALKANES [J].

ROLLA, F .

JOURNAL OF ORGANIC CHEMISTRY, 1981, 46 (19) :3909-3911

← 1 2 3 4 →